SCHEMBL18354527

SCHEMBL18354527

CCN(C(=O)c1ccc(C(F)(F)F)cc1)c1cccc(C(=O)Nc2c(Cl)cc(C(F)(C(F)(F)F)C(F)(F)F)cc2OC(F)F)c1F

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 10/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
MRGPRX4 Q96LA9 6/20 0.35
TLR7 Q9NYK1 1/20 0.34
SCN8A Q9UQD0 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18354405 0.95 DHODH (0.38) DHODHTAS1R3TAS1R1TAS1R2
SCHEMBL18354699 0.94 DHODH (0.37) DHODHTAS1R3TAS1R1TAS1R2
SCHEMBL18354199 0.94 DHODH (0.38) DHODHTAS1R3TAS1R1TAS1R2
SCHEMBL17482156 0.93 DHODH (0.37) DHODHTAS1R3TAS1R1TAS1R2
SCHEMBL18354050 0.93 DHODH (0.37) DHODHTAS1R3TAS1R1TAS1R2
SCHEMBL18354718 0.92 TAS1R3 (0.39) DHODHTAS1R3TAS1R1TAS1R2MRGPRX4
SCHEMBL18354398 0.91 MLYCD (0.39) DHODH
SCHEMBL18360165 0.91 DHODH (0.38) DHODHTAS1R3TAS1R1TAS1R2MRGPRX4
SCHEMBL18354645 0.91 HDAC8 (0.34) DHODHSCN8ASCN10A
SCHEMBL18354196 0.91 MAPT (0.37) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210051955-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2021-02-25 US disclosed
US-20180077930-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2018-03-22 US disclosed
US-20180077930-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2018-03-22 US disclosed
US-9839216-B2 Insecticidal compounds SYNGENTA PARTICIPATIONS AG (CH) 2017-12-12 US disclosed
US-9839216-B2 Insecticidal compounds SYNGENTA PARTICIPATIONS AG (CH) 2017-12-12 US disclosed
US-20170000120-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2017-01-05 US disclosed
US-20170000120-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2017-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180077930-A1 INSECTICIDAL COMPOUNDS ACHE, CYP4X1, ITPR3 DHODH 3024/4885TAS1R3 381/4885TAS1R1 817/4885
US-20210051955-A1 INSECTICIDAL COMPOUNDS ACHE, CYP4X1, ITPR3 DHODH 3024/4885TAS1R3 381/4885TAS1R1 817/4885
US-20170000120-A1 INSECTICIDAL COMPOUNDS ACHE, HDAC6, TUBA3C DHODH 3226/4885TAS1R3 455/4885TAS1R1 1016/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.