SCHEMBL18360640

SCHEMBL18360640

Cc1cc(C2NNC3=C2CN(C(=O)NC2CC(C)CN(Cc4cc5ccccc5n4C)C2)CC3)ccn1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.40
MCHR1 Q99705 1/20 0.38
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
CCR8 P51685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18360668 0.85 PRMT5 (0.35) FAAHPRMT5WDR77
SCHEMBL18360717 0.81 MAPK1 (0.45)
SCHEMBL15065565 0.80 PIP5K1C (0.45)
SCHEMBL18360599 0.80 FAAH (0.39) FAAHMCHR1
SCHEMBL807475 0.78 FAAH (0.40) FAAHMCHR1CCR8
SCHEMBL18360586 0.76 PKM (0.37)
SCHEMBL18360685 0.73 MAPK1 (0.44)
SCHEMBL18360718 0.72 MAPK1 (0.40)
SCHEMBL18360605 0.72 MAPK1 (0.46)
SCHEMBL18360672 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2615916-B1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS MERCK SHARP & DOHME (US) 2017-01-04 EP disclosed