SCHEMBL807475

SCHEMBL807475

Cc1cc(C(=N)C2=C(N)CCN(C(=O)NC3CC(C)CN(Cc4cc5ccccc5n4C)C3)C2)ccn1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.40
MCHR1 Q99705 1/20 0.38
CCR8 P51685 1/20 0.32
ACKR3 P25106 2/20 0.32
PROKR1 Q8TCW9 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807646 0.82 FAAH (0.38) FAAH
SCHEMBL18360599 0.78 FAAH (0.39) FAAHMCHR1
SCHEMBL18360640 0.78 FAAH (0.40) FAAHMCHR1CCR8
SCHEMBL15065565 0.78 PIP5K1C (0.45)
SCHEMBL15084329 0.66 FAAH (0.51) FAAHMCHR1HCRTR1HCRTR2
SCHEMBL15065068 0.64 PIP5K1C (0.44)
SCHEMBL18360666 0.63 ROCK2 (0.44)
SCHEMBL15065414 0.62
SCHEMBL15065500 0.62
SCHEMBL12073932 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed