SCHEMBL1838591

SCHEMBL1838591

COC(=O)c1c(F)cc(OCC(C2CCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)cc1F

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 2/20 0.32
CNR1 P21554 1/20 0.32
REN P00797 1/20 0.32
FPR1 P21462 2/20 0.31
FPR2 P25090 1/20 0.31
NR1H4 Q96RI1 4/20 0.31
CYP2C9 P11712 2/20 0.31
HSP90B1 P14625 1/20 0.31
PTGDR Q13258 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
KCNH2 Q12809 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1839025 0.93 LMNA (0.32) LMNATP53MAPTCNR1REN
SCHEMBL1840368 0.90 NR1H4 (0.33) LMNATP53MAPTNR1H4CYP2C9
SCHEMBL1841265 0.87 BACE1 (0.36) NR1H4
SCHEMBL1842508 0.86 GLA (0.43) LMNATP53PTGDRPTGDR2MEN1
SCHEMBL1843050 0.86 NR1H4 (0.33) LMNATP53MAPTCNR1REN
SCHEMBL1842591 0.86 NR1H4 (0.34) LMNATP53MAPTNR1H4CYP2C9
SCHEMBL1839912 0.86 NR1H4 (0.33) LMNATP53MAPTCNR1REN
SCHEMBL1840349 0.85 NR1H4 (0.40) LMNATP53MAPTCNR1REN
SCHEMBL1837605 0.85 ALDH1A1 (0.43) CNR1NR1H4CYP2C9CYP3A4MEN1
SCHEMBL1840310 0.85 NR1H4 (0.36) MAPTNR1H4CYP2C9PTGDRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed