SCHEMBL1840331

SCHEMBL1840331

O=C(NCc1ccccc1)C(C1CCCC1)C1(c2ccc(Cl)cc2)Nc2cc(F)c(F)cc2N1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.42
HPGD P15428 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CTSD P07339 1/20 0.40
CPB2 Q96IY4 1/20 0.39
KLK7 P49862 1/20 0.38
MMP1 P03956 1/20 0.38
FCER2 P06734 1/20 0.38
ADAM17 P78536 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
MDM2 Q00987 1/20 0.38
OGT O15294 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1842066 0.96 OPRL1 (0.39) CTSDADAM17SCN5ASCN9AMDM2
SCHEMBL4040798 0.91 EPHX1 (0.47) EPHX1HPGDNPC1RAB9ACPB2
SCHEMBL1840250 0.83 TP53 (0.36) NPC1RAB9AMDM2
SCHEMBL1838714 0.82 TP53 (0.38) EPHX1NPC1RAB9AMDM2
SCHEMBL4035029 0.81 NR1H4 (0.47) EPHX1HPGDNPC1RAB9A
SCHEMBL4040844 0.81 NR1H4 (0.47) EPHX1HPGDNPC1RAB9A
SCHEMBL1839859 0.81 AGER (0.37) MDM2
SCHEMBL4043373 0.80 CTSD (0.36) EPHX1CTSD
SCHEMBL1838873 0.79 SLC6A3 (0.42) MDM2
SCHEMBL3655058 0.79 NR1H4 (0.54) EPHX1NPC1RAB9AKLK7MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed