Prochlorperazine

Prochlorperazine

SCHEMBL18429

CN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Prochlorperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 9/20 1.00
MAPT P10636 7/20 1.00
MAPK1 P28482 7/20 1.00
ADRA2A P08913 7/20 1.00
ADRA2C P18825 7/20 1.00
SLC6A2 P23975 7/20 1.00
HTR2A P28223 7/20 1.00
SLC6A4 P31645 7/20 1.00
HRH1 P35367 7/20 1.00
DRD3 P35462 7/20 1.00
LMNA P02545 6/20 1.00
TP53 P04637 6/20 1.00
CYP3A4 P08684 6/20 1.00
SMN1; SMN2 Q16637 6/20 1.00
HTR1A P08908 6/20 1.00
ADRA1A P35348 6/20 1.00
SLC6A3 Q01959 6/20 1.00
KCNH2 Q12809 6/20 1.00
ADRA2B P18089 6/20 1.00
HTR2C P28335 6/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prochlorperazine SCHEMBL29358207 1.00 DRD2 (1.00) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL14126977 1.00 DRD2 (1.00) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL29369439 1.00 DRD2 (1.00) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL133595 0.99 DRD2 (0.98) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL2506559 0.99 DRD2 (0.98) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL1041250 0.99 DRD2 (0.98) DRD2MAPTMAPK1ADRA2AADRA2C
Perphenazine SCHEMBL28086447 0.94 MAPT (0.91) DRD2MAPTMAPK1ADRA2AADRA2C
Perphenazine SCHEMBL5307579 0.94 MAPT (0.91) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL10891828 0.93 MAPT (0.90) DRD2MAPTMAPK1ADRA2AADRA2C
SCHEMBL13485632 0.93 MAPT (0.86) DRD2MAPTMAPK1ADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 27471 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624036-B2 Method of treating post-traumatic stress disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
US-12624037-B2 Method of treating agitation, aggressive behavior, and impulse control disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
CN-122028919-A Compositions and methods for treating cancer by affecting cancer cell membrane receptors and exosomes derived therefrom 黄奇英 2026-05-12 CN claimed
WO-2026090164-A1 COMPOSITIONS COMPRISING ELISMETREP AND A SECOND THERAPEUTIC AGENT FOR TREATING OR PREVENTING MIGRAINE OR PAIN KALLYOPE, INC. (US) 2026-04-30 WO claimed
US-20260090584-A1 SYSTEMS AND METHODS FOR ESTIMATING AEROSOLIZATION EMISSION SCIENTIFIC HORIZONS CONSULTING LLC (US) 2026-04-02 US claimed
US-12577255-B2 MDM2-based modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-03-17 US claimed
EP-4704832-A2 BIFUNCTIONAL SMALL MOLECULES TO TARGET THE SELECTIVE DEGRADATION OF CIRCULATING PROTEINS Biohaven Therapeutics Ltd. (VG) 2026-03-11 EP claimed
EP-4698530-A1 NK3 MODULATORS AND USES THEREOF Kallyope, Inc. (US) 2026-02-25 EP claimed
US-20260034065-A1 EXTENDED RELEASE PHARMACEUTICAL FORMULATION DOUGLAS PHARMACEUTICALS LTD (NZ) 2026-02-05 US claimed
US-20260022117-A1 COMPOUNDS AND METHODS FOR THE ENHANCED DEGRADATION OF TARGETED PROTEINS ARVINAS OPERATIONS INC (US) 2026-01-22 US claimed
WO-1985003937-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1985-09-12 WO claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
US-4536403-A WITH CARISOPRODOL ROOKS J F GIRARD 1985-08-20 US claimed
EP-0126684-A2 Drug delivery system utilizing thermosetting gels MERCK & CO. INC. (US) 1984-11-28 EP claimed
US-4474752-A DIAMINE MODIFIED POLYOXYETHYLENE-POLYOXYPROPYLENE COPOLYMER MERCK & CO., INC. (US) 1984-10-02 US claimed
US-4407800-A TRYPANOCIDES UNIVERSITY OF VIRGINIA ALUMNI PATENTS FOUNDATION (US) 1983-10-04 US claimed
US-4334526-A Method for administering a dissociative, unconscious type of anesthesia HAMACHER EDWARD N 1982-06-15 US claimed
US-4246894-A Method and system for administering a dissociative, unconscious type of anesthesia HAMACHER EDWARD N 1981-01-27 US claimed
US-4175119-A Composition and method to prevent accidental and intentional overdosage with psychoactive drugs PORTER GARRY L 1979-11-20 US claimed
US-4111203-A OSMOTIC SYSTEM WITH MEANS FOR IMPROVING DELIVERY KINETICS OF SYSTEM ALZA CORPORATION (US) 1978-09-05 US claimed