Prochlorperazine

Prochlorperazine

SCHEMBL29358207

CN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Prochlorperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 9/20 1.00
MAPT P10636 7/20 1.00
MAPK1 P28482 7/20 1.00
ADRA2A P08913 7/20 1.00
ADRA2C P18825 7/20 1.00
SLC6A2 P23975 7/20 1.00
HTR2A P28223 7/20 1.00
SLC6A4 P31645 7/20 1.00
HRH1 P35367 7/20 1.00
DRD3 P35462 7/20 1.00
LMNA P02545 6/20 1.00
TP53 P04637 6/20 1.00
CYP3A4 P08684 6/20 1.00
SMN1; SMN2 Q16637 6/20 1.00
HTR1A P08908 6/20 1.00
ADRA1A P35348 6/20 1.00
SLC6A3 Q01959 6/20 1.00
KCNH2 Q12809 6/20 1.00
ADRA2B P18089 6/20 1.00
HTR2C P28335 6/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prochlorperazine SCHEMBL14126977 1.00 DRD2 (1.00) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL29369439 1.00 DRD2 (1.00) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL18429 1.00 DRD2 (1.00) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL133595 0.99 DRD2 (0.98) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL2506559 0.99 DRD2 (0.98) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL1041250 0.99 DRD2 (0.98) DRD2MAPTMAPK1ADRA2AADRA2C
Perphenazine SCHEMBL28086447 0.94 MAPT (0.91) DRD2MAPTMAPK1ADRA2AADRA2C
Perphenazine SCHEMBL5307579 0.94 MAPT (0.91) DRD2MAPTMAPK1ADRA2AADRA2C
Prochlorperazine SCHEMBL10891828 0.93 MAPT (0.90) DRD2MAPTMAPK1ADRA2AADRA2C
SCHEMBL13485632 0.93 MAPT (0.86) DRD2MAPTMAPK1ADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240277636-A1 COMBINATION COMPRISING AT LEAST ONE SEROTONIN REUPTAKE INHIBITOR AND AT LEAST ONE STIMULATOR OF POTASSIUM-CHLORIDE COTRANSPORTER TYPE 2 AND ITS MEDICAL USE UNIVERSITé LAVAL (CA) 2024-08-22 US claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
EP-4358947-A1 COMBINATION COMPRISING AT LEAST ONE SEROTONIN REUPTAKE INHIBITOR AND AT LEAST ONE STIMULATOR OF POTASSIUM-CHLORIDE COTRANSPORTER TYPE 2 AND ITS MEDICAL USE UNIVERSITE DE BORDEAUX (FR) 2024-05-01 EP claimed
CN-117897147-A Combination comprising at least one serotonin reuptake inhibitor and at least one potassium chloride type 2 cotransporter stimulator and medical use thereof 波尔多大学 2024-04-16 CN claimed
US-11672866-B2 Osteotropic nanoparticles for prevention or treatment of bone metastases UNM RAINFOREST INNOVATIONS 2023-06-13 US claimed
WO-2022268738-A1 COMBINATION COMPRISING AT LEAST ONE SEROTONIN REUPTAKE INHIBITOR AND AT LEAST ONE STIMULATOR OF POTASSIUM-CHLORIDE COTRANSPORTER TYPE 2 AND ITS MEDICAL USE Universite de Bordeaux (FR) 2022-12-29 WO claimed
US-12550235-B2 2026-02-10 US disclosed
US-20260034303-A1 Needle Assisted Injection Device Having Reduced Trigger Force ANTARES PHARMA, INC. (US) 2026-02-05 US disclosed
US-20250381149-A1 CATIONIC AMPHIPHILIC COMPOUND-BASED NANOPARTICLE COMPOSITIONS UNIVERSITEIT GENT (BE) 2025-12-18 US disclosed
US-20250276066-A1 METHODS, COMPOSITIONS AND COMPOUNDS FOR TREATING AGE-RELATED DISEASES AND CONDITIONS GERO PTE LTD (SG) 2025-09-04 US disclosed
US-20250262268-A1 Methods and Compositions for Inhibiting Viral Infection NEW YORK UNIVERSITY 2025-08-21 US disclosed
EP-4547229-A1 CATIONIC AMPHIPHILIC COMPOUND-BASED NANOPARTICLE COMPOSITIONS Universiteit Gent (BE) 2025-05-07 EP disclosed
WO-2025076082-A1 PEPTIDE NANOSPONGES FOR DRUG DELIVERY UNIVERSITY OF KANSAS (US) 2025-04-10 WO disclosed
WO-2022219021-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR TREATING REFRACTORY EPILEPSY INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2022-10-20 WO disclosed
WO-2022219021-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR TREATING REFRACTORY EPILEPSY INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2022-10-20 WO disclosed
US-20220330396-A1 MICROWAVE HEATING UNIT AND METHOD JT INTERNATIONAL SA (CH) 2022-10-13 US disclosed
WO-2022175673-A1 PROCHLORPERAZINE FOR USE IN THE TREATMENT OF NEUROBLASTOMA HEALX LIMITED (GB) 2022-08-25 WO disclosed
WO-2022173333-A2 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING AGE-RELATED DISEASES AND CONDITIONS GERO PTE. LTD. (SG) 2022-08-18 WO disclosed
EP-4011396-A1 RELEASABLE CONJUGATES QuiaPEG Pharmaceuticals AB (SE) 2022-06-15 EP disclosed
EP-3747289-B1 MICROWAVE HEATING UNIT AND METHOD NVX LABS GMBH (CH) 2022-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260034303-A1 Needle Assisted Injection Device Having Reduced Trigger Force TIMM44, SARAF, TIMM50 DRD2 2480/4885MAPT 1680/4885MAPK1 1511/4885
US-11672866-B2 Osteotropic nanoparticles for prevention or treatment of bone metastases SOST, ACP3, KLK3 DRD2 3763/4885MAPT 3975/4885MAPK1 2477/4885
US-20250381149-A1 CATIONIC AMPHIPHILIC COMPOUND-BASED NANOPARTICLE COMPOSITIONS NPC1L1, NPC1, ABCB4 DRD2 4816/4885MAPT 2743/4885MAPK1 4537/4885
US-12550235-B2 MTX2, CRY2, MTX1 DRD2 4116/4885MAPT 883/4885MAPK1 2213/4885
US-20250276066-A1 METHODS, COMPOSITIONS AND COMPOUNDS FOR TREATING AGE-RELATED DISEASES AND CONDITIONS UPF1, NLN, BRCA1 DRD2 4318/4885MAPT 523/4885MAPK1 1254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.