SCHEMBL18436553

SCHEMBL18436553

CSc1cnc2c(C)cccc2c1C1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
TNF P01375 1/20 0.36
LITAF Q99732 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
PDK2 Q15119 3/20 0.35
PDK4 Q16654 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
PDK1 Q15118 1/20 0.33
PARP14 Q460N5 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19012578 0.84 PARP1 (0.40) PARP1TNFLITAFHTR1AADRA1D
SCHEMBL19012437 0.78 TNF (0.40) PARP1TNFLITAFHTR1AADRA1D
SCHEMBL18436735 0.75 TNF (0.38) PARP1TNFLITAFHTR1AADRA1D
SCHEMBL18436773 0.74 PARP1 (0.40) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL16951638 0.73 MAP3K14 (0.37) HTR1AMEN1RAB9AKMT2ALMNA
SCHEMBL21336609 0.72 HTR1A (0.39) PARP1TNFLITAFHTR1AADRA1D
SCHEMBL16959393 0.66 ALDH1A1 (0.46) CYP1A2CYP2A6
SCHEMBL862479 0.65 CCR1 (0.68) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL19000956 0.65 PDK2 (0.33) PARP1PDK2PDK4KDM4EPDK1
SCHEMBL19012433 0.63 PARP1 (0.44) PARP1HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed