SCHEMBL18436773

SCHEMBL18436773

CSc1cnc2c(C)cccc2c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.40
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CRHR1 P34998 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE7A Q13946 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18436374 0.82 AXL (0.46) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL7494879 0.76 HAVCR2 (0.52) PARP1MEN1KMT2ANPC1RAB9A
SCHEMBL18436553 0.74 PARP1 (0.36) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL9652797 0.71 ATP4A (0.50)
SCHEMBL2020438 0.70 KMT2A (0.71) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL442075 0.70 HAVCR2 (0.46) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL862479 0.70 CCR1 (0.68) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL12093642 0.69 MAPT (0.40) MEN1KMT2ANPC1RAB9ACYP1A2
SCHEMBL31523701 0.68 HTR1A (0.45) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL24507816 0.67 CYP2A6 (0.41) PARP1HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed