SCHEMBL18436657

SCHEMBL18436657

CC1CN(c2ccc(I)cc2)CC(C)N1C(=O)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43
RBP4 P02753 1/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
KLF5 Q13887 1/20 0.41
NAMPT P43490 1/20 0.39
SLC6A7 Q99884 1/20 0.39
PDE10A Q9Y233 1/20 0.39
ALDH1A1 P00352 1/20 0.39
RIPK1 Q13546 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18436805 0.89 SMN1; SMN2 (0.50) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL19012370 0.89 SMN1; SMN2 (0.50) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL18436815 0.85 CSF1R (0.46) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL19001092 0.85 PLA2G1B (0.51) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL19001032 0.85 PLA2G1B (0.51) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL19012742 0.85 HSD11B1 (0.46) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL19012534 0.85 HSD11B1 (0.46) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL21336587 0.77 ALDH1A1 (0.46) HSD11B1SMN1; SMN2CHRNB2CHRNB4CHRNA3
SCHEMBL20750442 0.74 CHRNB2 (0.61) HSD11B1L3MBTL1SMN1; SMN2CHRNB2CHRNB4
SCHEMBL20690378 0.69 L3MBTL1 (0.67) L3MBTL1SMN1; SMN2CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed