SCHEMBL1845259

SCHEMBL1845259

Cc1cn(-c2ccc([N+](=O)[O-])cc2)cn1.O=[N+]([O-])c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.51
HTT P42858 1/20 0.46
KMT2A Q03164 3/20 0.45
MAPT P10636 2/20 0.44
HSPB1 P04792 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PTGS1 P23219 1/20 0.42
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1037500 0.93 HTT (0.51) POLBHTTKMT2AMAPTCYP1A2
SCHEMBL18754697 0.84 CYP3A4 (0.56) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL17632850 0.77 HTR2A (0.58) POLBMAPTHSPB1PTGS1ALDH1A1
SCHEMBL23292585 0.76 TLR2 (0.49) KMT2AALDH1A1LMNA
SCHEMBL1617550 0.76 ALDH1A1 (0.47) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL27985278 0.76 CYP1A2 (0.65) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL6756946 0.75 FGFR1 (0.50) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL2470937 0.75 PTGS2 (0.45) POLBKMT2AMAPTCYP1A2CYP3A4
SCHEMBL22465893 0.74 HTR2A (0.42) POLBHTTKMT2AMAPTCYP1A2
SCHEMBL2253987 0.74 TSHR (0.38) POLBMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2315588-A1 6-1H-IMIDAZO-QUINAZOLINE AND QUINOLINES DERIVATIVES, NEW MAO INHIBITORS AND IMIDAZOLINE RECEPTOR LIGANDS Rottapharm S.p.A. (IT) 2011-05-04 EP disclosed