SCHEMBL18486174

SCHEMBL18486174

Nc1ccnc(-c2cc(F)cc(CCCN3CCCC3)c2)c1N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 2/20 0.48
DRD2 P14416 2/20 0.48
SLC6A4 P31645 1/20 0.48
MAP4K4 O95819 4/20 0.41
HRH3 Q9Y5N1 3/20 0.40
MAPK13 O15264 3/20 0.39
MAPK12 P53778 3/20 0.39
MAPK11 Q15759 3/20 0.39
MAPK14 Q16539 3/20 0.39
EHMT2 Q96KQ7 1/20 0.38
EHMT1 Q9H9B1 1/20 0.38
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
SCN5A Q14524 1/20 0.37
LTA4H P09960 1/20 0.36
HTR1A P08908 1/20 0.36
DRD1 P21728 1/20 0.36
DRD5 P21918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18474444 0.82 SLC6A3 (0.48) SLC6A3DRD2SLC6A4MAP4K4HRH3
SCHEMBL17555897 0.81 LTA4H (0.46) MAP4K4HRH3MEN1LMNAHTT
SCHEMBL18482037 0.79 SLC6A3 (0.56) SLC6A3DRD2SLC6A4MAP4K4HRH3
SCHEMBL18486943 0.78 NOS1 (0.46) MAP4K4
SCHEMBL18476441 0.77 SLC6A3 (0.47) SLC6A3DRD2SLC6A4MAP4K4HRH3
SCHEMBL3873265 0.72 EHMT2 (0.44) SLC6A3DRD2SLC6A4HRH3EHMT2
SCHEMBL17555820 0.68 KDM1A (0.42)
SCHEMBL18487394 0.68 ADORA2A (0.36) MEN1KMT2A
SCHEMBL18474439 0.68 SLC6A3 (0.60) SLC6A3DRD2SLC6A4HRH3LMNA
SCHEMBL17555600 0.68 CLK2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023972-A1 3-(1H-IMIDAZO[4,5-C]PYRIDIN-2-YL)-1H-PYRAZOLO[4,3-B]PYRIDINES AND THERAPEUTIC USES THEREOF SAMUMED, LLC. (US) 2017-02-09 WO disclosed