SCHEMBL18488359

SCHEMBL18488359

Cc1ccc2ncc(Cl)c(CO)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
TNF P01375 3/20 0.42
MAPK1 P28482 1/20 0.40
HTR1A P08908 2/20 0.40
ADRA1D P25100 2/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
PKM P14618 1/20 0.39
PARP1 P09874 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37
PLAT P00750 1/20 0.37
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18450619 0.81 TNF (0.45) LMNATNFMAPK1CYP2C9CYP2C19
SCHEMBL9380208 0.78 LMNA (0.50) LMNATNFMAPK1HTR1AADRA1D
SCHEMBL5042933 0.77 PKM (0.42) LMNATNFMAPK1HTR1AADRA1D
SCHEMBL440082 0.75 LMNA (0.47) LMNATNFHTR1AADRA1DADRA1A
SCHEMBL18449197 0.74 TNF (0.60) TNFCYP2C9CYP2C19
SCHEMBL11061888 0.72 KDM4E (0.42) LMNAMAPK1HTR1AADRA1DADRA1A
SCHEMBL27413106 0.71 HTR1A (0.37) LMNATNFMAPK1HTR1AADRA1D
SCHEMBL1029308 0.70 LMNA (0.36) LMNATNFMAPK1HTR1AADRA1D
SCHEMBL13074891 0.69 PLG (0.43) LMNATNFMAPK1HTR1APKM
SCHEMBL9724121 0.69 LMNA (0.62) LMNAMAPK1HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023905-A1 HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF TNF ALPHA BRISTOL-MYERS SQUIBB COMPANY (US) 2017-02-09 WO disclosed