SCHEMBL1850454

SCHEMBL1850454

O=C(Nc1cccc(-c2cccc3cc(C(O)c4cccc(C(F)(F)F)c4)sc23)c1)c1cccc(-c2cccc3cc(C(O)c4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
GPR52 Q9Y2T5 3/20 0.51
KCNK3 O14649 2/20 0.47
MAPK1 P28482 1/20 0.46
LMNA P02545 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
PTGS1 P23219 1/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
BRAF P15056 2/20 0.45
KCNK9 Q9NPC2 1/20 0.44
PDGFRB P09619 1/20 0.44
KDR P35968 1/20 0.44
LCK P06239 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TYMS P04818 1/20 0.43
P2RX1 P51575 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3198656 0.87 GPR52 (0.49) GPR52MEN1KMT2ARAB9AALDH1A1
SCHEMBL3219110 0.86 GPR52 (0.51) GPR52BRAF
SCHEMBL3209079 0.86 GPR52 (0.70) GPR52ALDH1A1POLB
SCHEMBL3198211 0.85 GPR52 (0.70) GPR52ALDH1A1POLB
SCHEMBL3218871 0.84 GPR52 (0.71) GPR52ALDH1A1POLB
SCHEMBL1850455 0.83 GPR52 (0.49) GPR52MEN1KMT2ARAB9AALDH1A1
SCHEMBL1849541 0.82 GPR52 (0.66) GPR52HTTALDH1A1POLB
SCHEMBL3204669 0.82 GPR52 (0.49) MAPTGPR52MEN1KMT2ARAB9A
SCHEMBL1850259 0.80 GPR52 (0.61) GPR52ALDH1A1POLB
SCHEMBL1850452 0.79 GPR52 (0.46) MAPTGPR52RAB9ABRAFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed