SCHEMBL1850452

SCHEMBL1850452

NC(=O)c1cccc(-c2cccc3cc(C(OC(=O)c4cccc(-c5cccc6cc(C(O)c7cccc(C(F)(F)F)c7)sc56)c4)c4cccc(C(F)(F)F)c4)sc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 8/20 0.46
S1PR4 O95977 1/20 0.38
S1PR5 Q9H228 1/20 0.38
SCD O00767 1/20 0.36
CES2 O00748 1/20 0.36
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PLG P00747 1/20 0.34
PLAU P00749 1/20 0.34
PLAT P00750 1/20 0.34
DHODH Q02127 1/20 0.34
SLC9A1 P19634 1/20 0.34
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3219110 0.92 GPR52 (0.51) GPR52S1PR4S1PR5SCDCES2
SCHEMBL1851846 0.90 GPR52 (0.45) GPR52S1PR4S1PR5SCDCES2
SCHEMBL1850455 0.89 GPR52 (0.49) GPR52S1PR4S1PR5SCDCES2
SCHEMBL1850259 0.86 GPR52 (0.61) GPR52S1PR4S1PR5SCDALDH1A1
SCHEMBL1861066 0.85 GPR52 (0.64) GPR52S1PR4S1PR5SCDALDH1A1
SCHEMBL3204669 0.84 GPR52 (0.49) GPR52S1PR4S1PR5SCDCES2
SCHEMBL3198656 0.84 GPR52 (0.49) GPR52S1PR4S1PR5SCDCES2
SCHEMBL3198211 0.80 GPR52 (0.70) GPR52S1PR4S1PR5SCDALDH1A1
SCHEMBL1852537 0.80 GPR52 (0.45) GPR52S1PR4S1PR5SCDCES2
SCHEMBL1850454 0.79 MAPT (0.52) GPR52ALDH1A1MAPTRAB9ABRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed