SCHEMBL1851797

SCHEMBL1851797

CCCCCOc1ccc(C#Cc2ccc(C[N+]([O-])(CC(=O)O)Cc3ccc(C(F)(F)F)cc3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.43
PTGES O14684 2/20 0.43
PPARG P37231 2/20 0.43
PLA2G4B P0C869 1/20 0.42
ACACB O00763 4/20 0.42
S1PR4 O95977 2/20 0.41
S1PR1 P21453 2/20 0.41
S1PR3 Q99500 2/20 0.41
S1PR5 Q9H228 1/20 0.41
PSEN1 P49768 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
FAAH O00519 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
PPARA Q07869 1/20 0.40
FFAR1 O14842 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1851799 0.84 ACACB (0.44) ALOX5PTGESPPARGPLA2G4BACACB
SCHEMBL1856893 0.82 ALOX5 (0.42) ALOX5PTGESPPARGPLA2G4BACACB
SCHEMBL5045341 0.79 PPARA (0.44) PPARGPLA2G4BACACBS1PR4S1PR1
SCHEMBL1851802 0.77 PTGES (0.44) ALOX5PTGESPPARGACACBS1PR1
SCHEMBL1853816 0.76 PTGES (0.43) ALOX5PTGESPPARGPLA2G4BACACB
SCHEMBL5039929 0.74 S1PR2 (0.49) ACACBS1PR1S1PR3FAAH
SCHEMBL6023332 0.74 NR5A1 (0.42) PLA2G4BACACBS1PR1FAAHTP53
SCHEMBL28423723 0.73 NR5A1 (0.56) PLA2G4BTP53TSHRPPARA
SCHEMBL1855304 0.73 ACACB (0.42) PTGESACACBFAAH
SCHEMBL1852713 0.73 ACACB (0.51) ACACBFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470102-B1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) MERCK SERONO SA (CH) 2011-05-25 EP disclosed