SCHEMBL18529092

SCHEMBL18529092

O=C1COc2ncc(Cl)nc2N1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.32
AKR1B1 P15121 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
NR3C2 P08235 3/20 0.31
MGLL Q99685 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384794 0.80 MAPK1 (0.32) KCNH2CYP11B1CYP11B2NR3C2
SCHEMBL31057602 0.78 KCNH2 (0.32) KCNH2
SCHEMBL18529102 0.78 KCNH2 (0.32) KCNH2
SCHEMBL31057590 0.76 KCNH2 (0.30) KCNH2
SCHEMBL18529063 0.76 KCNH2 (0.30) KCNH2
SCHEMBL18542847 0.76 NR3C2 (0.34) KCNH2NR3C2
SCHEMBL16651977 0.73 MMP12 (0.33) CYP11B1CYP11B2NR3C2
SCHEMBL21429876 0.72 KCNH2 (0.39) KCNH2NR3C2
SCHEMBL30306227 0.72 KCNH2 (0.39) KCNH2NR3C2
SCHEMBL30406269 0.72 KCNH2 (0.35) KCNH2NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724427-A1 A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF Bugworks Research, Inc. (US) 2026-04-15 EP disclosed
WO-2024252423-A1 A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF BUGWORKS RESEARCH INDIA PVT LTD (IN) 2024-12-12 WO disclosed
EP-3717490-B1 ANTI-BACTERIAL HETEROCYCLIC COMPOUNDS AND THEIR SYNTHESIS BUGWORKS RES INC (US) 2023-05-24 EP disclosed
EP-3717490-B1 ANTI-BACTERIAL HETEROCYCLIC COMPOUNDS AND THEIR SYNTHESIS BUGWORKS RES INC (US) 2023-05-24 EP disclosed
US-11590142-B2 Oxazolidinone antibiotic compounds and process of preparation Bugworks Research, Inc. (US) 2023-02-28 US disclosed
EP-3774790-B1 OXAZOLIDINONE ANTIBIOTIC COMPOUNDS AND PROCESS OF PREPARATION BUGWORKS RES INC (US) 2023-01-25 EP disclosed
EP-3774790-B1 OXAZOLIDINONE ANTIBIOTIC COMPOUNDS AND PROCESS OF PREPARATION BUGWORKS RES INC (US) 2023-01-25 EP disclosed
EP-3634968-B1 HETEROCYCLIC COMPOUNDS USEFUL AS ANTI-BACTERIAL AGENTS AND METHOD FOR PRODUCTION THEREOF BUGWORKS RES INC (US) 2023-01-25 EP disclosed
EP-3634968-B1 HETEROCYCLIC COMPOUNDS USEFUL AS ANTI-BACTERIAL AGENTS AND METHOD FOR PRODUCTION THEREOF BUGWORKS RES INC (US) 2023-01-25 EP disclosed
US-11401277-B2 Anti-bacterial heterocyclic compounds and their synthesis Bugworks Research, Inc. (US) 2022-08-02 US disclosed
US-20190270755-A1 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-09-05 US disclosed
US-20190270755-A1 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-09-05 US disclosed
US-10364254-B2 Compounds for use in antibacterial applications GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-07-30 US disclosed
US-10364254-B2 Compounds for use in antibacterial applications GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-07-30 US disclosed
US-20190031680-A1 COMPOUNDS FOR US IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-01-31 US disclosed
US-20190031680-A1 COMPOUNDS FOR US IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-01-31 US disclosed
WO-2018225097-A1 HETEROCYCLIC COMPOUNDS USEFUL AS ANTI-BACTERIAL AGENTS AND METHOD FOR PRODUCTION THEREOF BUGWORKS RESEARCH INDIA PVT LTD (IN) 2018-12-13 WO disclosed
EP-3334739-A2 ANTIBACTERIAL AGENTS COMPRISING A PYRAZINO[2,3-B][1,4]OXAZIN-3-ONE OR A RELATED RING SYSTEM GlaxoSmithKline Intellectual Property Development Limited (GB) 2018-06-20 EP disclosed
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed
WO-2017029602-A2 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190270755-A1 COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS MRPL21, CFTR, NRDC KCNH2 2823/4885AKR1B1 3853/4885CYP11B1 4652/4885
US-11401277-B2 Anti-bacterial heterocyclic compounds and their synthesis HLA-B, BAX, REN KCNH2 3099/4885AKR1B1 392/4885CYP11B1 10/4885
US-11590142-B2 Oxazolidinone antibiotic compounds and process of preparation ALPI, OXA1L, ALPL KCNH2 4322/4885AKR1B1 598/4885CYP11B1 39/4885
US-20190031680-A1 COMPOUNDS FOR US IN ANTIBACTERIAL APPLICATIONS CFTR, MRPL21, CLPP KCNH2 2998/4885AKR1B1 4327/4885CYP11B1 4802/4885
US-10364254-B2 Compounds for use in antibacterial applications MRPL21, CFTR, NRDC KCNH2 2823/4885AKR1B1 3853/4885CYP11B1 4652/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.