SCHEMBL1853992

SCHEMBL1853992

CCCCCCCCCCCCNC(=O)c1ccc(CN(Cc2ccc(C(F)(F)F)nc2)C(=O)C(=O)O)cc1.CCCCCCCCCCCCNC(=O)c1ccc(CN(Cc2ccc(S(C)(=O)=O)cc2)C(=O)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.46
MLYCD O95822 1/20 0.44
EPHX2 P34913 7/20 0.41
NAAA Q02083 2/20 0.41
TMEM97 Q5BJF2 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
NAMPT P43490 1/20 0.40
PTGS2 P35354 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
OPRK1 P41145 1/20 0.40
NR1H4 Q96RI1 1/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1855106 0.95 MLYCD (0.49) CA2MLYCDNAAATMEM97SIGMAR1
SCHEMBL1855672 0.89 CA2 (0.57) CA2MLYCDEPHX2NAAATMEM97
SCHEMBL1850884 0.85 NAAA (0.44) CA2MLYCDNAAATMEM97SIGMAR1
SCHEMBL5047490 0.83 MLYCD (0.53) CA2MLYCDNAAATMEM97SIGMAR1
SCHEMBL1853427 0.82 TMEM97 (0.56) CA2MLYCDEPHX2NAAATMEM97
SCHEMBL1852987 0.82 TMEM97 (0.56) CA2MLYCDEPHX2NAAATMEM97
SCHEMBL1854307 0.80 NAAA (0.48) CA2NAAATMEM97SIGMAR1NAMPT
SCHEMBL1853434 0.80 TMEM97 (0.53) CA2MLYCDNAAATMEM97SIGMAR1
SCHEMBL27601057 0.79 MLYCD (0.55) CA2MLYCDNAAAL3MBTL1NAMPT
SCHEMBL1857574 0.78 NAAA (0.57) CA2MLYCDNAAATMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470102-B1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) MERCK SERONO SA (CH) 2011-05-25 EP claimed