SCHEMBL185405

SCHEMBL185405

Cc1ccccc1C(CC(N)=O)C(C)C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NR3C2 P08235 2/20 0.39
PTGER3 P43115 1/20 0.39
ESR1 P03372 1/20 0.37
ACP3 P15309 1/20 0.37
CTSA P10619 4/20 0.35
TAAR1 Q96RJ0 1/20 0.35
CYP2C19 P33261 3/20 0.35
GLS O94925 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363392 0.82 NR3C2 (0.47) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL29048166 0.80 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ANPSR1NR3C2
SCHEMBL11088063 0.80 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL14108456 0.80 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL29998155 0.79 ALDH1A1 (0.42) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL185647 0.77 TAAR1 (0.57) ALDH1A1LMNANPSR1TAAR1CYP2C19
SCHEMBL185424 0.76 ALDH1A1 (0.42) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL18181442 0.76 TAAR1 (0.55) ESR1TAAR1CYP1A2CYP3A4
SCHEMBL185645 0.73 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL3668722 0.73 ALDH1A1 (0.45) ALDH1A1KMT2AMAPTNR3C2PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401260-A1 DIOXO-IMIDAZOLIDINE DERIVATIVES, WHICH INHIBIT THE ENZYME SOAT-1, AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING THEM Galderma Research & Development (FR) 2012-01-04 EP disclosed
WO-2010097465-A1 DIOXO-IMIDAZOLIDINE DERIVATIVES, WHICH INHIBIT THE ENZYME SOAT-1, AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING THEM GALDERMA RESEARCH & DEVELOPMENT (FR) 2010-09-02 WO disclosed