SCHEMBL18543791

SCHEMBL18543791

C[C@@]1(O)CC[C@]2(Cc3ccc(Br)cc3C2)C(=O)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.36
PARP1 P09874 1/20 0.35
CMA1 P23946 1/20 0.34
AHR P35869 1/20 0.34
BRD4 O60885 1/20 0.34
METAP1 P53582 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
BACE1 P56817 3/20 0.32
HSD11B1 P28845 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9958538 0.81 TDP2 (0.46) TDP2PARP1CMA1AHRBRD4
SCHEMBL9959281 0.79 BACE1 (0.40) TDP2PARP1CMA1AHRBRD4
SCHEMBL18065482 0.77 PNMT (0.38) TDP2CMA1AHRBRD4METAP1
SCHEMBL18065483 0.77 PNMT (0.38) TDP2CMA1AHRBRD4METAP1
SCHEMBL10249815 0.77 CA1 (0.42) TDP2PARP1CMA1AHRBRD4
SCHEMBL9948406 0.77 CA1 (0.42) TDP2PARP1CMA1AHRBRD4
SCHEMBL9947977 0.77 CA1 (0.42) TDP2PARP1CMA1AHRBRD4
SCHEMBL9958466 0.73 BACE1 (0.40) TDP2CMA1AHRMETAP1CA1
SCHEMBL31076 0.73 BACE1 (0.40) TDP2CMA1AHRMETAP1CA1
SCHEMBL9958457 0.73 TDP2 (0.41) TDP2PARP1CMA1AHRBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655378-B1 COMPOUNDS AND THEIR USE AS BACE INHIBITORS ASTRAZENECA AB (SE) 2017-03-01 EP disclosed