SCHEMBL1854575

SCHEMBL1854575

O=S(=O)(Oc1cccc2oc(Cc3cccc(C(F)(F)F)c3)nc12)C(F)(F)F.Oc1cccc2oc(Cc3cccc(C(F)(F)F)c3)nc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.42
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
RAB9A P51151 5/20 0.38
NPC1 O15118 3/20 0.38
POLB P06746 3/20 0.38
APLNR P35414 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
PTPRC P08575 1/20 0.35
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPN6 P29350 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1858526 0.95 MAPT (0.39) HTR2BKMT2AMAPTTDP1RAB9A
SCHEMBL1857128 0.86 HTR2B (0.47) HTR2BKMT2AMAPTTDP1RAB9A
SCHEMBL3198348 0.73 MAOB (0.40) HTR2B
SCHEMBL1854688 0.72 ACSL1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1848465 0.71 MAOB (0.38) HTR2BKMT2AMAPTTDP1
SCHEMBL1855792 0.70 GPR52 (0.51) KMT2AMAPTTDP1RAB9ANPC1
SCHEMBL1852090 0.65 TP53 (0.36)
SCHEMBL18409661 0.65 RXRA (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL27725812 0.65 TP53 (0.47) KMT2AMAPTSMN1; SMN2CYP1A2CYP2C9
SCHEMBL1848567 0.63 ALOX5 (0.56) HTR2BKMT2AMAPTTDP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed