SCHEMBL18554143

SCHEMBL18554143

COC(=O)CC[C@@H](Cc1ccc(-c2ccccc2)cc1)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MME P08473 2/20 0.47
MAOB P27338 1/20 0.42
HDAC1 Q13547 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42
PPARG P37231 4/20 0.42
PPARA Q07869 3/20 0.42
SRR Q9GZT4 1/20 0.41
PSAT1 Q9Y617 1/20 0.41
PTGES O14684 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18554144 1.00 MME (0.47) MMEMAOBHDAC1HDAC6PPARG
SCHEMBL18554221 0.86 PTGES (0.42) MMEPPARGPPARASRRPSAT1
SCHEMBL18554224 0.86 PTGES (0.42) MMEPPARGPPARASRRPSAT1
SCHEMBL18554199 0.85 FFAR1 (0.53) MMEPPARGPPARA
SCHEMBL18554201 0.85 FFAR1 (0.53) MMEPPARGPPARA
Hydrochloric Acid SCHEMBL18554214 0.84 FFAR1 (0.51) MMEPPARGPPARASRRPSAT1
Hydrochloric Acid SCHEMBL18554213 0.84 FFAR1 (0.51) MMEPPARGPPARASRRPSAT1
SCHEMBL18576599 0.81 MME (0.45) MMEHDAC1HDAC6PPARGPPARA
SCHEMBL18554285 0.79 ADRB1 (0.41) MMEALDH1A1MAPT
SCHEMBL18554307 0.79 ADRB1 (0.41) MMEALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017033128-A1 BIPHENYL-SUBSTITUED 4-AMINO-BUTYRIC ACID DERIVATIVES AND THEIR USE IN THE SYNTHESIS OF NEP INHIBITORS NOVARTIS AG (CH) 2017-03-02 WO disclosed
WO-2017033128-A1 BIPHENYL-SUBSTITUED 4-AMINO-BUTYRIC ACID DERIVATIVES AND THEIR USE IN THE SYNTHESIS OF NEP INHIBITORS NOVARTIS AG (CH) 2017-03-02 WO disclosed