SCHEMBL18558154

SCHEMBL18558154

CC(C)(C)N/C(=N/C(=O)c1cccc(Cl)c1)Nc1cc(-c2cccc(Cl)c2)n[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
ALPL P05186 1/20 0.39
CNR2 P34972 2/20 0.39
SLC6A2 P23975 2/20 0.38
CHRNA1 P02708 1/20 0.38
CHRNG P07510 1/20 0.38
ITGA5 P08648 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
SLC6A4 P31645 1/20 0.38
CHRNA3 P32297 1/20 0.38
CYP2C19 P33261 1/20 0.38
HRH1 P35367 1/20 0.38
CHRNA7 P36544 1/20 0.38
OPRK1 P41145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18558126 0.93 RAB9A (0.38) GRM5NPC1RAB9ABCHEACHE
SCHEMBL18558380 0.93 NPC1 (0.42) NPC1RAB9ABCHEACHEALPL
SCHEMBL18558387 0.93 RAF1 (0.41) GRM5NPC1RAB9ABCHEACHE
SCHEMBL18558596 0.92 RAF1 (0.42) GRM5RAF1ALDH1A1SMN1; SMN2
SCHEMBL18558156 0.91 MAPT (0.36) GRM5BCHEACHEALPLCNR2
SCHEMBL18558388 0.90 MAPT (0.39) GRM5BCHEACHEALPLCNR2
SCHEMBL18558653 0.90 IDO1 (0.39) NPC1RAB9AALPLSLC6A2CHRNA1
SCHEMBL18557825 0.90 ALPL (0.38) GRM5BCHEACHEALPLCNR2
SCHEMBL18558394 0.88 RAF1 (0.39) BCHEACHEALPLCNR2RAF1
SCHEMBL18558029 0.84 NPC1 (0.40) NPC1RAB9ABCHEACHEALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9580388-B2 Pyrazolyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2017-02-28 US disclosed