SCHEMBL1858459

SCHEMBL1858459

CC1CC(c2ccc(Cl)cc2)CC(C)(C)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.37
DRD2 P14416 1/20 0.37
KDM1A O60341 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37
CYP2D6 P10635 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
SRD5A1 P18405 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CCR2 P41597 1/20 0.35
SLC2A1 P11166 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MAP1LC3B Q9GZQ8 1/20 0.34
MAPK1 P28482 1/20 0.34
ADRB2 P07550 1/20 0.34
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23071529 0.82 IDH1 (0.39) CYP2C19MEN1KMT2AALDH1A1LMNA
SCHEMBL335898 0.82 ESR2 (0.52) CYP2C19ALDH1A1LMNACYP3A4
SCHEMBL28343291 0.82 ALDH1A1 (0.33) CYP2C19ALDH1A1LMNACYP3A4HTT
SCHEMBL11461120 0.79 ALDH1A1 (0.33) CYP2C19ALDH1A1LMNACYP3A4HTT
SCHEMBL11481127 0.79 MAPK1 (0.47) HTR3ASRD5A1CCR2SLC6A3MAP1LC3B
SCHEMBL1445179 0.78 HTR3A (0.45) HTR3ADRD2SRD5A1MEN1KMT2A
SCHEMBL19031705 0.78 LMNA (0.37) CYP2D6CYP2B6CYP2C19ALDH1A1LMNA
Bicarbonate SCHEMBL28346273 0.77 ESR2 (0.46) CYP2C19ALDH1A1LMNACYP3A4HTT
SCHEMBL23071549 0.77 IDH1 (0.40) CYP2C19ALDH1A1LMNACYP3A4HTT
SCHEMBL7784850 0.77 ALDH1A1 (0.37) CYP2C19MEN1KMT2AALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7939509-B2 Partial and full agonists of A1 adenosine receptors GILEAD SCIENCES, INC. (US) 2011-05-10 US disclosed