SCHEMBL1859508

SCHEMBL1859508

Nc1ccnc(N)c1-c1ccc(C(F)(F)F)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.41
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
KMT2A Q03164 1/20 0.40
RET P07949 1/20 0.40
KDM4E B2RXH2 1/20 0.39
CASP3 P42574 1/20 0.37
KDM1A O60341 1/20 0.36
MAOB P27338 1/20 0.36
PTGS1 P23219 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
PDE2A O00408 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RECQL P46063 1/20 0.35
FEN1 P39748 4/20 0.35
ALOX5AP P20292 3/20 0.35
DHFR P00374 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29595709 0.75 NPSR1 (0.53) KIF11NPSR1KMT2AKDM4ECASP3
SCHEMBL811160 0.75 NPSR1 (0.53) KIF11NPSR1KMT2AKDM4ECASP3
SCHEMBL2934747 0.74 KIF11 (0.43) KIF11NPSR1KMT2AKDM4EKDM1A
SCHEMBL6033597 0.72 CASP3 (0.45) KIF11NOS3NOS2NPSR1KMT2A
SCHEMBL28510482 0.71 CYP11B1 (0.43) KIF11NPSR1KMT2AKDM4EKDM1A
SCHEMBL31114170 0.71 CYP11B1 (0.43) KIF11NPSR1KMT2AKDM4EKDM1A
Ammonia Solution, Strong SCHEMBL1863056 0.70 MAPT (0.40) KIF11NOS3NOS2NPSR1KMT2A
SCHEMBL27344645 0.70 KIF11 (0.63) KIF11NPSR1KMT2AKDM4ECASP3
SCHEMBL1862303 0.70 KIF11 (0.41) KIF11NPSR1KMT2AKDM4ECASP3
SCHEMBL10416583 0.70 KMT2A (0.41) KIF11NPSR1KMT2AKDM4EKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed