SCHEMBL18599183

SCHEMBL18599183

CC(C)[C@H](CC#N)c1cc(Br)ccc1OCC#N

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.38
ALDH1A1 P00352 3/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 3/20 0.33
TSHR P16473 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
AAK1 Q2M2I8 2/20 0.32
CYSLTR2 Q9NS75 1/20 0.32
CYSLTR1 Q9Y271 1/20 0.32
CCR5 P51681 1/20 0.31
RAB9A P51151 2/20 0.30
NPC1 O15118 1/20 0.30
LMNA P02545 1/20 0.30
CSNK2A1 P68400 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9918207 1.00 TP53 (0.38) TP53ALDH1A1HTTSMN1; SMN2MAPT
SCHEMBL9918824 0.91 HPGD (0.39) TP53ALDH1A1HTTSMN1; SMN2MAPT
SCHEMBL9918202 0.86 TRPV4 (0.36)
SCHEMBL9918206 0.85 LMNA (0.38) ALDH1A1HTTSMN1; SMN2MAPTTSHR
SCHEMBL9921720 0.85 TP53 (0.40) TP53ALDH1A1HTTSMN1; SMN2MAPT
SCHEMBL12251263 0.85 ALDH1A1 (0.33) ALDH1A1HTTSMN1; SMN2MAPTHPGD
SCHEMBL13678297 0.84
SCHEMBL171764 0.81 SGMS2 (0.34) ALDH1A1MEN1KMT2ALMNA
SCHEMBL16691093 0.80 TP53 (0.38) TP53ALDH1A1HTTSMN1; SMN2MAPT
SCHEMBL19062265 0.79 TP53 (0.37) TP53ALDH1A1HTTSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2348023-B9 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors INCYTE HOLDINGS CORP (US) 2017-03-08 EP disclosed