SCHEMBL18599280

SCHEMBL18599280

OOc1cncc(OCC2CCOCC2)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.47
RIPK2 O43353 1/20 0.41
CHRNB2 P17787 3/20 0.40
CHRNA4 P43681 3/20 0.40
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
XDH P47989 1/20 0.38
SLC2A1 P11166 1/20 0.38
KDM4C Q9H3R0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3108687 0.85 CHRNB4 (0.55) CYP11B2RIPK2CHRNB2CHRNA4CHRNB4
SCHEMBL3103772 0.82 CHRNB2 (0.52) CYP11B2RIPK2CHRNB2CHRNA4KDM4E
SCHEMBL15716470 0.81 CYP11B2 (0.45) CYP11B2RIPK2CHRNB2CHRNA4CHRNB4
Lithium SCHEMBL29705636 0.74 CYP11B2 (0.45) CYP11B2RIPK2CHRNB2CHRNA4KDM4E
SCHEMBL12525730 0.72 SLC2A1 (0.46) XDHSLC2A1KDM4C
SCHEMBL13096931 0.72 CYP2D6 (0.39) CYP11B2CHRNB4CHRNA3CYP2D6XDH
SCHEMBL19405964 0.72 CHRNB4 (0.61) CHRNB2CHRNA4CHRNB4CHRNA3KDM4E
SCHEMBL13097262 0.71 CHRNB4 (0.46) CYP11B2CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4909692 0.71 PIK3CA (0.44) CYP2D6XDH
SCHEMBL29136349 0.70 DHFR (0.40) CYP11B2CYP2D6XDHSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2920183-B1 THIENO[3,2-C]PYRIDIN-4(5H)-ONES AS BET INHIBITORS GLAXOSMITHKLINE LLC (US) 2017-03-08 EP disclosed