SCHEMBL18599596

SCHEMBL18599596

FC(F)(F)c1cncc2cccc(I)c12

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.37
CYP11B1 P15538 3/20 0.37
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ERN1 O75460 1/20 0.32
AXL P30530 1/20 0.32
CYP17A1 P05093 1/20 0.32
SCN9A Q15858 1/20 0.31
ULK1 O75385 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18495140 0.79 ELANE (0.40) CYP11B2CYP11B1KDM4EALDH1A1MAPT
SCHEMBL17228307 0.79 CYP3A4 (0.42) CYP11B2CYP11B1KDM4EALDH1A1MAPT
SCHEMBL18477492 0.77 CYP11B2 (0.36) CYP11B2CYP11B1KDM4EALDH1A1MAPT
SCHEMBL18848566 0.77 PDPK1 (0.34) KDM4EALDH1A1
SCHEMBL18599581 0.76 ROCK2 (0.35) CYP11B2CYP11B1
SCHEMBL11142241 0.73 CYP11B2 (0.55) CYP11B2CYP11B1KDM4EALDH1A1MAPT
SCHEMBL17228312 0.72 TDP1 (0.42) KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL17228308 0.72 SLC22A12 (0.37) CYP11B2CYP11B1CYP17A1
SCHEMBL18599582 0.72 AHR (0.35) KDM4EALDH1A1MAPT
SCHEMBL18599583 0.72 ROCK2 (0.37) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138843-A1 ISOQUINOLINESULFONYL DERIVATIVE AS RHO KINASE INHIBITOR Medshine Discovery Inc. (CN) 2017-03-08 EP disclosed