SCHEMBL18599581

SCHEMBL18599581

Fc1cncc2cccc(I)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 2/20 0.35
PLK4 O00444 1/20 0.35
NQO2 P16083 1/20 0.35
MARK3 P27448 1/20 0.35
MAP2K3 P46734 1/20 0.35
CDK9 P50750 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKCD Q05655 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PKN1 Q16512 1/20 0.35
PKN2 Q16513 1/20 0.35
MARK2 Q7KZI7 1/20 0.35
MAP4K3 Q8IVH8 1/20 0.35
AURKB Q96GD4 1/20 0.35
PRKD2 Q9BZL6 1/20 0.35
TAOK3 Q9H2K8 1/20 0.35
PDPK1 O15530 1/20 0.32
CYP11B1 P15538 2/20 0.30
CYP11B2 P19099 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18848566 0.81 PDPK1 (0.34) PDPK1
SCHEMBL18495139 0.78 ACHE (0.39) ROCK2ROCK1PLK4NQO2MARK3
SCHEMBL24672067 0.76 ALDH1A1 (0.41) PDPK1
SCHEMBL998210 0.76 CYP3A4 (0.46) ROCK2ROCK1PLK4NQO2MARK3
SCHEMBL18599582 0.76 AHR (0.35) PDPK1
SCHEMBL18599583 0.76 ROCK2 (0.37) ROCK2ROCK1PLK4MARK3PRKCD
SCHEMBL18599596 0.76 CYP11B2 (0.37) CYP11B1CYP11B2
SCHEMBL18599597 0.76
SCHEMBL28644536 0.73 ROCK2 (0.47) ROCK2ROCK1PLK4NQO2MARK3
SCHEMBL14308389 0.72 ROCK2 (0.36) ROCK2ROCK1PLK4NQO2MARK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138843-A1 ISOQUINOLINESULFONYL DERIVATIVE AS RHO KINASE INHIBITOR Medshine Discovery Inc. (CN) 2017-03-08 EP disclosed