SCHEMBL18600520

SCHEMBL18600520

CC(=O)N1CCN(c2ccccc2Br)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
HPGD P15428 2/20 0.54
USP2 O75604 1/20 0.54
TP53 P04637 1/20 0.54
MAPK1 P28482 1/20 0.54
KMT2A Q03164 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
MEN1 O00255 2/20 0.51
LMNA P02545 2/20 0.51
MAPT P10636 2/20 0.51
HTT P42858 1/20 0.51
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
NCF1 P14598 2/20 0.50
TSHR P16473 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
SMO Q99835 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30937462 1.00 ALDH1A1 (0.59) ALDH1A1HPGDUSP2TP53MAPK1
SCHEMBL113679 0.84 ALDH1A1 (0.55) ALDH1A1HPGDUSP2MAPK1KMT2A
SCHEMBL5919531 0.84 ALDH1A1 (0.61) ALDH1A1HPGDUSP2TP53MAPK1
SCHEMBL27926749 0.81 MGLL (0.46) ALDH1A1HPGDMAPK1KMT2ASMN1; SMN2
SCHEMBL28235242 0.81 MGLL (0.46) ALDH1A1HPGDMAPK1KMT2ASMN1; SMN2
SCHEMBL9565829 0.81 AKR1C3 (0.62) ALDH1A1HPGDUSP2TP53MAPK1
SCHEMBL3436305 0.81 ALDH1A1 (0.76) ALDH1A1KMT2AHTTNCF1TSHR
SCHEMBL3801245 0.81 GAA (0.65) ALDH1A1KMT2ASMN1; SMN2MEN1LMNA
SCHEMBL30062550 0.80 GPR119 (0.52) ALDH1A1TP53KMT2ASMN1; SMN2MEN1
SCHEMBL1928396 0.80 GPR119 (0.52) ALDH1A1TP53KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926286-B2 Vortioxetine intermediate and synthesis process thereof SHANGHAI SYNCORES TECHNOLOGIES INC. LTD. (CN) 2018-03-27 US disclosed
US-9926286-B2 Vortioxetine intermediate and synthesis process thereof SHANGHAI SYNCORES TECHNOLOGIES INC. LTD. (CN) 2018-03-27 US disclosed
US-20170088530-A1 NEW VORTIOXETINE INTERMEDIATE AND SYNTHESIS PROCESS THEREOF SHANGHAI SYNCORES TECHNOLOGIES INC. LTD. (CN) 2017-03-30 US disclosed
US-20170088530-A1 NEW VORTIOXETINE INTERMEDIATE AND SYNTHESIS PROCESS THEREOF SHANGHAI SYNCORES TECHNOLOGIES INC. LTD. (CN) 2017-03-30 US disclosed
EP-3141543-A1 NEW VORTIOXETINE INTERMEDIATE AND SYNTHESIS PROCESS THEREOF Shanghai Syncores Technologies, Inc. (CN) 2017-03-15 EP disclosed
CN-100400523-C Substituted piperazines, (1,4) diaza * class and 2, 5-diazabicyclo (2.2.1) heptanes as histamine H1 and/or H3 antagonists or histamine H3 reverse antagonists GLAXO GROUP LTD (GB) 2008-07-09 CN disclosed
CN-101070309-A Substituted piperazines as histamine H1 and/or H3 antagonists or histamine H3 reverse antagonists, (1, 4) diazabi and 2, 5-diazabicyclo (2.2.1) heptanes GLAXO GROUP LTD (GB) 2007-11-14 CN disclosed
CN-1726201-A Substituted piperazines, (1,4) diaza * class and 2, 5-diazabicyclo (2.2.1) heptanes as histamine H1 and/or H3 antagonists or histamine H3 reverse antagonists GLAXO GROUP LTD (GB) 2006-01-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170088530-A1 NEW VORTIOXETINE INTERMEDIATE AND SYNTHESIS PROCESS THEREOF CYP3A4, CYP4B1, COMT ALDH1A1 249/4885HPGD 1270/4885USP2 1848/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.