SCHEMBL18614902

SCHEMBL18614902

N#Cc1[c]nncc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.39
MAPK1 P28482 1/20 0.39
METAP2 P50579 1/20 0.39
NPSR1 Q6W5P4 4/20 0.37
ALDH1A1 P00352 4/20 0.37
TDP1 Q9NUW8 1/20 0.37
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
GABRA5 P31644 3/20 0.36
GABRA3 P34903 3/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
KDM4E B2RXH2 4/20 0.34
HPGD P15428 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
GABRA1 P14867 2/20 0.34
HSD17B10 Q99714 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1551998 0.73 AXL (0.36) MAPK1ALDH1A1GABRG2GABRB3GABRA5
SCHEMBL10806706 0.66 CHEK1 (0.41) L3MBTL1MAPK1METAP2NPSR1ALDH1A1
SCHEMBL5664674 0.64 L3MBTL1 (0.39) L3MBTL1MAPK1NPSR1ALDH1A1ADORA2A
SCHEMBL1227720 0.63 KMT2A (0.46) L3MBTL1MAPK1NPSR1ALDH1A1TDP1
SCHEMBL12825464 0.63 ALDH1A1 (0.46) L3MBTL1MAPK1NPSR1ALDH1A1GABRG2
SCHEMBL7220037 0.63 ADORA1 (0.49) L3MBTL1MAPK1NPSR1ALDH1A1ADORA2A
SCHEMBL6971354 0.63 L3MBTL1 (0.38) L3MBTL1MAPK1NPSR1ALDH1A1TDP1
SCHEMBL1146097 0.63 CYP1A2 (0.57) L3MBTL1NPSR1ALDH1A1TDP1GABRG2
SCHEMBL7213782 0.62 NPSR1 (0.53) L3MBTL1MAPK1NPSR1ALDH1A1TDP1
Bromide SCHEMBL20536256 0.61 ALDH1A1 (0.51) L3MBTL1MAPK1NPSR1ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3347097-A1 SUBSTITUTED HETEROARYL COMPOUNDS AND METHODS OF USE Sunshine Lake Pharma Co., Ltd. (CN) 2018-07-18 EP claimed
WO-2017044434-A1 SUBSTITUTED HETEROARYL COMPOUNDS AND METHODS OF USE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2017-03-16 WO claimed