SCHEMBL18616366

SCHEMBL18616366

CCc1ccc2c(c1)CCCC2N

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 8/20 0.47
KDM4C Q9H3R0 2/20 0.42
ACHE P22303 2/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16543139 1.00 OPRD1 (0.47) OPRD1KDM4CACHEESR1ESR2
SCHEMBL16543141 1.00 OPRD1 (0.47) OPRD1KDM4CACHEESR1ESR2
SCHEMBL14606247 0.90 DRD2 (0.42) OPRD1ACHEESR1ESR2
SCHEMBL13499147 0.87 OPRD1 (0.47) OPRD1ACHEESR1ESR2
SCHEMBL6330755 0.87 ACHE (0.50) OPRD1ACHE
SCHEMBL8281689 0.87 ACHE (0.50) OPRD1ACHE
Hydrochloric Acid SCHEMBL3171185 0.85 ACHE (0.49) OPRD1ACHE
SCHEMBL1726880 0.83 OPRD1 (0.45) OPRD1ACHEESR1ESR2
SCHEMBL4517111 0.83 OPRD1 (0.45) OPRD1ACHEESR1ESR2
SCHEMBL1726878 0.83 OPRD1 (0.45) OPRD1ACHEESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017040449-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE BRISTOL-MYERS SQUIBB COMPANY (US) 2017-03-09 WO disclosed