SCHEMBL18616784

SCHEMBL18616784

CCc1ccc2c(c1)CCNC2C

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOA P21397 8/20 0.51
DRD2 P14416 2/20 0.51
TSHR P16473 2/20 0.51
HSD17B10 Q99714 2/20 0.51
KDM4E B2RXH2 2/20 0.51
CYP2C9 P11712 1/20 0.51
DRD3 P35462 1/20 0.51
HIF1A Q16665 1/20 0.51
DRD4 P21917 1/20 0.51
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KDM1A O60341 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21335646 0.87 MAOA (0.49) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL20884606 0.87 MAOA (0.51) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL20672036 0.83 MAOA (0.47) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL25920451 0.80 ADRB2 (0.55) DRD2KDM4EDRD4KDM1AGAA
SCHEMBL20883964 0.78 KDM1A (0.47) DRD2KDM4EDRD4KDM1AGAA
SCHEMBL7820935 0.77 MAOA (0.56) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL1009166 0.76 ALDH1A1 (0.48) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL24529091 0.76 CYP4F2 (0.47) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL22680298 0.76 MAOA (0.54) MAOADRD2TSHRHSD17B10KDM4E
SCHEMBL21959060 0.76 MAOA (0.64) MAOADRD2TSHRHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017205193-A1 SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS USEFUL AS GPR120 AGONISTS MERCK SHARP & DOHME CORP. (US) 2017-11-30 WO disclosed
WO-2017040449-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE BRISTOL-MYERS SQUIBB COMPANY (US) 2017-03-09 WO disclosed