SCHEMBL18622355

SCHEMBL18622355

FCc1ccc(-n2nnnc2-c2c(-c3cc(Cl)ccc3Cl)nc3ccccn23)cc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1I3 Q14994 17/20 0.47
ALDH1A1 P00352 1/20 0.40
NR1I2 O75469 2/20 0.40
DPP4 P27487 1/20 0.39
LMNA P02545 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14740335 0.91 LMNA (0.46) NR1I3ALDH1A1NR1I2DPP4LMNA
SCHEMBL14740306 0.87 NR1I3 (0.45) NR1I3ALDH1A1DPP4LMNAHSD17B10
SCHEMBL14740449 0.85 NR1I3 (0.45) NR1I3ALDH1A1DPP4LMNAHSD17B10
SCHEMBL18622357 0.84 P2RX7 (0.41) NR1I3ALDH1A1LMNAHSD17B10CYP1A2
SCHEMBL14739184 0.83 ALDH1A1 (0.50) NR1I3ALDH1A1NR1I2DPP4LMNA
SCHEMBL18622362 0.83 NR1I3 (0.44) NR1I3ALDH1A1NR1I2DPP4CYP1A2
SCHEMBL14745122 0.78 KCNN4 (0.42) NR1I3ALDH1A1NR1I2DPP4
SCHEMBL14739635 0.78 L3MBTL1 (0.44) ALDH1A1LMNAHSD17B10
SCHEMBL14740234 0.76 ALDH1A1 (0.43) NR1I3ALDH1A1LMNAHSD17B10CYP1A2
SCHEMBL14740387 0.75 DPP4 (0.42) NR1I3ALDH1A1NR1I2DPP4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9593109-B2 Bicyclic agonists of GPR131 and uses thereof CYMABAY THERAPEUTICS, INC. (US) 2017-03-14 US disclosed