SCHEMBL18645758

SCHEMBL18645758

Cc1cc(C(C)(C)C)cc(-c2ccc(Cl)cc2)c1O

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
POLB P06746 1/20 0.38
RXRB P28702 1/20 0.37
CNR1 P21554 2/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4366547 0.85 HSP90AA1 (0.49) CYP1A2CYP2C9CYP2C19MEN1KMT2A
SCHEMBL17500060 0.82 ESR2 (0.47) ALOX5PTGS1PTGS2CYP1A2CYP2C9
SCHEMBL19732817 0.79 GABRA1 (0.50) CYP1A2CYP2C9CYP2C19MEN1KMT2A
SCHEMBL28121289 0.77 ALDH1A1 (0.52) ALOX5MEN1KMT2AAKR1C2AKR1C1
SCHEMBL31720848 0.77 POLB (0.42) MEN1KMT2APOLBCNR1
SCHEMBL15674488 0.76 NPSR1 (0.40) CYP1A2CYP2C9CYP2C19MEN1KMT2A
SCHEMBL17500122 0.76 HDAC4 (0.47) ALOX5MEN1KMT2AESR1ESR2
SCHEMBL3672236 0.75 CA2 (0.55) ALOX5PTGS1PTGS2CYP1A2CYP2C9
SCHEMBL18645759 0.72 KIF11 (0.54) ALOX5PTGS1PTGS2CYP1A2CYP2C9
SCHEMBL201609 0.72 GABRA1 (0.57) CYP1A2CYP2C9CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017044889-A1 LRH-1 MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-03-16 WO disclosed