SCHEMBL18650482

SCHEMBL18650482

O=NN1CCc2cc(C3CCc4ccccc4N3N=O)ccc2C1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 6/20 0.34
TSHR P16473 1/20 0.33
SIGMAR1 Q99720 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 2/20 0.31
HTR6 P50406 2/20 0.31
CHRM4 P08173 2/20 0.31
HTR7 P34969 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
SRD5A1 P18405 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554586 0.77 TSHR (0.40) TSHRDRD4DRD3CHRM4CHRM2
SCHEMBL31327521 0.72 MAOA (0.52) TSHRDRD4DRD3MAPTMEN1
SCHEMBL1025209 0.72 MAOA (0.52) TSHRDRD4DRD3MAPTMEN1
SCHEMBL20847929 0.67 MAOA (0.53) DRD4DRD3
SCHEMBL19035881 0.67 MAOA (0.49) SIGMAR1DRD4DRD3HTR6HTR7
SCHEMBL21020950 0.66 HTR2C (0.33) HSD17B3TSHRSIGMAR1DRD3HTR6
SCHEMBL1530624 0.65 ABHD6 (0.44) HSD17B3
SCHEMBL28415182 0.63 NOTUM (0.43) HSD17B3MAPTMEN1KMT2A
SCHEMBL20854483 0.59 HTR2A (0.42) HSD17B3HTR7SRD5A1
SCHEMBL11623429 0.59 ALDH1A1 (0.39) MAPTSRD5A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017045648-A1 PREPARATION METHOD FOR DEUTERATED COMPOUND 正大天晴药业集团股份有限公司 2017-03-23 WO disclosed