SCHEMBL18657152

SCHEMBL18657152

CC(=O)OCC#Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.45
MAPT P10636 6/20 0.44
ALDH1A1 P00352 4/20 0.44
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
THRB P10828 1/20 0.43
CYP2C9 P11712 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAOB P27338 1/20 0.43
PTPN2 P17706 1/20 0.42
PTPN1 P18031 1/20 0.42
PTPN6 P29350 1/20 0.42
PTPN11 Q06124 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30401530 0.87 MAPT (0.42) MAPK1MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL31348837 0.86 ALDH1A1 (0.47) MAPTALDH1A1SMN1; SMN2LMNACYP1A2
SCHEMBL6696133 0.83 ALDH1A1 (0.51) MAPTALDH1A1TP53SMN1; SMN2LMNA
SCHEMBL75802 0.78 CYP2D6 (0.45) MAPTALDH1A1LMNACYP2D6HPGD
SCHEMBL7575151 0.76 CASP3 (0.40) MAPTALDH1A1SMN1; SMN2LMNACYP1A2
SCHEMBL31103292 0.76 MAPK1 (0.45) MAPK1MAPTALDH1A1MAOBMEN1
SCHEMBL10102348 0.75 CASP3 (0.47) MAPK1MAPTALDH1A1MEN1HSP90AA1
SCHEMBL6318644 0.75 TSHR (0.48) MAPTALDH1A1CYP2C19MEN1HSP90AA1
SCHEMBL8950594 0.75 ALDH1A1 (0.39) MAPTALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL15235706 0.74 POLB (0.54) MAPTALDH1A1PKMMAOBPTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558445-B1 INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PYRROLOBENZODIAZEPINES MEDIMMUNE LTD (GB) 2017-03-22 EP disclosed