SCHEMBL18667147

SCHEMBL18667147

CC(C)(C)OC(=O)NCc1cnc(N2CCNC(=O)CC2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.39
CRBN Q96SW2 3/20 0.36
DDB1 Q16531 2/20 0.36
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
GFER P55789 1/20 0.34
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
CA12 O43570 2/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
CKS1B P61024 1/20 0.33
SKP1 P63208 1/20 0.33
SKP2 Q13309 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
OGA O60502 1/20 0.33
PRMT5 O14744 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18667145 0.87 L3MBTL1 (0.42) L3MBTL1KDM4ELMNAGFERCA1
SCHEMBL18667310 0.82 LMNA (0.45) L3MBTL1KDM4ELMNAALDH1A1MAPK1
SCHEMBL18667020 0.82 TDP1 (0.44) L3MBTL1KDM4ELMNA
SCHEMBL21250387 0.80 CKS1B (0.41) L3MBTL1KDM4ELMNAGFERCA1
SCHEMBL18667058 0.80 CKS1B (0.41) L3MBTL1GFERCA1CA2CA9
SCHEMBL21939563 0.78 HRH3 (0.44) L3MBTL1GFERSIRT2SIRT1SIRT3
SCHEMBL18667148 0.78 EIF2AK4 (0.35) CRBNLMNAALDH1A1
SCHEMBL26759389 0.77 PIK3CA (0.41) LMNAALDH1A1MAPK1
SCHEMBL20493701 0.75 ALDH1A1 (0.35) CRBNLMNAALDH1A1MAPK1OGA
Hydrochloric Acid SCHEMBL20493992 0.73 OGA (0.39) LMNAALDH1A1MAPK1OGA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240025890-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES INC (US) 2024-01-25 US disclosed
US-11814376-B2 Hepatitis b core protein modulators ASSEMBLY BIOSCIENCES, INC. (US) 2023-11-14 US disclosed
US-20230044112-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2023-02-09 US disclosed
US-10968211-B2 Hepatitis B core protein modulators ASSEMBLY BIOSCIENCES, INC. (US) 2021-04-06 US disclosed
EP-3782626-A1 HEPATITIS B CORE PROTEIN MODULATORS Assembly Biosciences, Inc. (US) 2021-02-24 EP disclosed
US-20200131168-A1 HEPATITIS B CORE PROTEIN MODULATORS INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION 2020-04-30 US disclosed
WO-2017048950-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2017-03-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240025890-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS L3MBTL1 1920/4885CRBN 777/4885DDB1 226/4885
US-20230044112-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS L3MBTL1 1920/4885CRBN 777/4885DDB1 226/4885
US-10968211-B2 Hepatitis B core protein modulators HAVCR2, FABP1, MAVS L3MBTL1 1920/4885CRBN 777/4885DDB1 226/4885
US-11814376-B2 Hepatitis b core protein modulators HAVCR2, FABP1, MAVS L3MBTL1 1920/4885CRBN 777/4885DDB1 226/4885
US-20200131168-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS L3MBTL1 1920/4885CRBN 777/4885DDB1 226/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.