SCHEMBL18683051

SCHEMBL18683051

COC(=O)C[C@](C)(NC(=O)OC(C)(C)C)c1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
AKT1 P31749 2/20 0.37
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
SCN9A Q15858 1/20 0.36
AAK1 Q2M2I8 2/20 0.36
CA12 O43570 2/20 0.36
CA14 Q9ULX7 2/20 0.36
CA1 P00915 1/20 0.36
CA7 P43166 1/20 0.36
GUCY1B2 O75343 2/20 0.36
GUCY1A2 P33402 2/20 0.36
GUCY1A1 Q02108 2/20 0.36
GUCY1B1 Q02153 2/20 0.36
IDO1 P14902 1/20 0.35
DRD2 P14416 1/20 0.35
SSTR4 P31391 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21677304 1.00 LMNA (0.40) LMNAPOLBCTSSCTSKAKT1
SCHEMBL21677273 0.89 NLRP3 (0.42) LMNAPOLBCTSSCTSKAKT1
SCHEMBL4665018 0.84 LMNA (0.39) LMNAPOLBCTSSCTSKAKT1
SCHEMBL4665019 0.84 AKT1 (0.39) LMNAPOLBCTSSCTSKAKT1
SCHEMBL31486571 0.78 AAK1 (0.32) LMNAPOLBAKT1MTNR1AMTNR1B
SCHEMBL31486781 0.78 DRD2 (0.32) LMNAPOLBAAK1CA12CA14
SCHEMBL31486754 0.77 SMN1; SMN2 (0.36) POLBCTSSCTSKAAK1SMN1; SMN2
SCHEMBL18683500 0.75 LMNA (0.39) LMNAPOLBCTSSCTSKAKT1
SCHEMBL20349827 0.75 BACE1 (0.40) LMNAGUCY1B2GUCY1A2GUCY1A1GUCY1B1
SCHEMBL18683050 0.74 LMNA (0.38) LMNAPOLBCTSSCTSKAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017050978-A1 2,3,4,5-TETRAHYDROPYRIDIN-6-AMINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2017-03-30 WO disclosed