SCHEMBL18686018

SCHEMBL18686018

CCOC(=O)C1CNCC2CC(=O)Nc3ccccc3N21

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.39
GAA P10253 2/20 0.38
NPC1 O15118 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 2/20 0.37
KMT2A Q03164 1/20 0.37
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
CASP3 P42574 1/20 0.37
CASP2 P42575 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2575403 0.76 HTR2A (0.62) ALDH1A1GAARAB9AKMT2ABRD4
SCHEMBL2575269 0.73 HTR2A (0.41) ALDH1A1KDM4EGAARAB9AKMT2A
SCHEMBL2572351 0.73 HTR2A (0.41) ALDH1A1KDM4EGAAKMT2ABRD4
SCHEMBL1420993 0.72 ALDH1A1 (0.63) ALDH1A1KDM4EHPGDGAANPC1
SCHEMBL27927982 0.69 NR1D1 (0.47) KDM4EHPGDLMNA
SCHEMBL1184927 0.68 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDGAAMAPK1
SCHEMBL30377419 0.67 PKM (0.46) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL692058 0.66 HTR2C (0.41) ALDH1A1KDM4EHPGDMAPK1SMN1; SMN2
SCHEMBL2014604 0.66 HTR2C (0.51) ALDH1A1KDM4EGAA
SCHEMBL693673 0.66 HTR2C (0.51) ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3150607-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF AbbVie Inc. (US) 2017-04-05 EP disclosed