SCHEMBL1869874

SCHEMBL1869874

O=S(=O)(Cl)C1CC(OCc2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
CTSK P43235 1/20 0.44
NAAA Q02083 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
EPHX2 P34913 1/20 0.40
OPRM1 P35372 2/20 0.40
OPRL1 P41146 2/20 0.40
DPP4 P27487 1/20 0.40
MMP9 P14780 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
TMEM97 Q5BJF2 1/20 0.38
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
PRMT8 Q9NR22 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
PDPK1 O15530 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25354547 0.85 OPRM1 (0.46) CTSLCTSBCTSKCA1CA2
SCHEMBL21885808 0.83 CA2 (0.49) CTSLCTSBCTSKNAAACA1
SCHEMBL20672954 0.83 CTSL (0.44) CTSLCTSBCTSKNAAACA1
SCHEMBL24815593 0.83 CA2 (0.49) CTSLCTSBCTSKNAAACA1
SCHEMBL1873174 0.83 CTSL (0.44) CTSLCTSBCTSKNAAAALDH1A1
SCHEMBL20595210 0.83 CTSL (0.44) CTSLCTSBCTSKNAAACA1
SCHEMBL24898491 0.82 CTSL (0.43) CTSLCTSBCTSKNAAACA1
SCHEMBL29260419 0.82 CTSL (0.43) CTSLCTSBCTSKNAAACA1
Potassium Ion SCHEMBL1868694 0.82 CTSL (0.43) CTSLCTSBCTSKNAAAALDH1A1
SCHEMBL1868696 0.82 CTSL (0.43) CTSLCTSBCTSKNAAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025103502-A1 COMPOUNDS AND METHODS OF TREATING CANCERS CULLGEN INC. (US) 2025-05-22 WO disclosed
WO-2023288254-A1 HETEROCYCLIC COMPOUNDS AS MAP4K1 INHIBITORS BLUEPRINT MEDICINES CORPORATION (US) 2023-01-19 WO disclosed
EP-2496575-B1 HETEROCYCLIC SULFONAMIDE DERIVATIVES USEFUL AS MEK INHIBITORS NOVARTIS AG (CH) 2014-04-30 EP disclosed
US-8466289-B2 Heterocyclic sulfonamide derivatives NOVARTIS AG (CH) 2013-06-18 US disclosed
US-8466289-B2 Heterocyclic sulfonamide derivatives NOVARTIS AG (CH) 2013-06-18 US disclosed
US-8466289-B2 Heterocyclic sulfonamide derivatives NOVARTIS AG (CH) 2013-06-18 US disclosed
EP-2496575-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES USEFUL AS MEK INHIBITORS Novartis AG (CH) 2012-09-12 EP disclosed
US-20110190334-A1 Heterocyclic Sulfonamide Derivatives NOVARTIS AG (CH) 2011-08-04 US disclosed
US-20110190334-A1 Heterocyclic Sulfonamide Derivatives NOVARTIS AG (CH) 2011-08-04 US disclosed
US-20110190334-A1 Heterocyclic Sulfonamide Derivatives NOVARTIS AG (CH) 2011-08-04 US disclosed
WO-2011054828-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES USEFUL AS MEK INHIBITORS NOVARTIS AG (CH) 2011-05-12 WO disclosed
WO-2011054828-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES USEFUL AS MEK INHIBITORS NOVARTIS AG (CH) 2011-05-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190334-A1 Heterocyclic Sulfonamide Derivatives BRAF, KSR2, NRAS CTSL 3558/4885CTSB 1022/4885CTSK 2893/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.