SCHEMBL18699192

SCHEMBL18699192

CCC(C)(C)c1cc(C(F)(F)F)c(/C(C)=C\C#N)cn1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.36
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
GABRB2 P47870 2/20 0.36
GABRB1 P18505 1/20 0.36
AR P10275 3/20 0.32
GAA P10253 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
LRRK2 Q5S007 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17808229 0.87 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL17808225 0.87 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL17813810 0.80 GABRA1 (0.42) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL16455580 0.80 GABRA1 (0.42) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL18699191 0.72 MAPT (0.37) ARGAAALDH1A1HPGDL3MBTL1
SCHEMBL17816233 0.65 CYP1A2 (0.41) ARGAAALDH1A1HPGDL3MBTL1
SCHEMBL17797764 0.64 GABRA1 (0.31) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL17808248 0.64 ASPH (0.33)
SCHEMBL17808249 0.64 PDE3B (0.35)
SCHEMBL18699194 0.63 IDO1 (0.41) ARALDH1A1L3MBTL1NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611248-B2 Chemical compounds SYNGENTA LIMITED (GB) 2017-04-04 US disclosed