SCHEMBL18767167

SCHEMBL18767167

CCCN(CCC)C(=O)c1cc(Cl)nc(OCc2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.43
PTGES O14684 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
ADORA1 P30542 1/20 0.42
APP P05067 1/20 0.41
GRM5 P41594 1/20 0.41
TP53 P04637 1/20 0.40
HTT P42858 1/20 0.40
LIMK1 P53667 1/20 0.39
LIMK2 P53671 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
RAF1 P04049 1/20 0.38
MAP2K1 Q02750 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18767170 0.86 ALOX5 (0.43) ALOX5PTGESMEN1KMT2AHPGD
SCHEMBL18767168 0.82 TSHR (0.39) ALDH1A1HPGDTP53HTTKDM4E
SCHEMBL731278 0.81 MEN1 (0.56) MEN1KMT2AHPGDGRM5TP53
SCHEMBL730969 0.79 LMNA (0.59) ALOX5PTGESMEN1KMT2AALDH1A1
SCHEMBL30931811 0.79 LMNA (0.59) ALOX5PTGESMEN1KMT2AALDH1A1
SCHEMBL18767173 0.78 PTGES (0.39) ALOX5PTGESMEN1KMT2AADORA3
SCHEMBL8894460 0.75 ALOX5 (0.63) ALOX5MEN1KMT2AALDH1A1HDAC1
SCHEMBL8894465 0.72 MEN1 (0.69) ALOX5MEN1KMT2AALDH1A1HPGD
SCHEMBL12076214 0.72 MEN1 (0.67) ALOX5PTGESMEN1KMT2AALDH1A1
SCHEMBL603696 0.71 NUDT1 (0.48) ALOX5PTGESALDH1A1GRM5HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017066742-A1 BACE-2 INHIBITORY COMPOUNDS AND RELATED METHODS OF USE JORTAN PHARMACEUTICALS INC. (US) 2017-04-20 WO disclosed