SCHEMBL1879639

SCHEMBL1879639

CSc1nccc(C=O)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 6/20 0.39
CCR1 P32246 1/20 0.39
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 4/20 0.35
HPGD P15428 2/20 0.35
ALOX15 P16050 1/20 0.35
PARP1 P09874 1/20 0.34
POLB P06746 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CCNT1 O60563 1/20 0.33
CCNA2 P20248 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17420132 0.80 MEN1 (0.40) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL4109091 0.77 HASPIN (0.37) KMT2ANPC1RAB9AALDH1A1CCR1
SCHEMBL23985444 0.76 MEN1 (0.43) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL28836041 0.76 L3MBTL1 (0.55) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL12273053 0.74 MEN1 (0.36) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL12273055 0.74 MEN1 (0.36) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL2563638 0.73 MAPK9 (0.41) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL29842006 0.73 KMT2A (0.41) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL1717209 0.72
SCHEMBL5045978 0.72 GPR84 (0.50) KMT2AMEN1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 353 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109824602-B Synthesis method of 4-chloro-2-methylthiopyrimidine 南京哈柏医药科技有限公司 2023-10-27 CN claimed
CN-116283793-A Synthesis process of 2-methylthio-4-chloro-5-bromopyrimidine 南京哈柏医药科技有限公司 2023-06-23 CN claimed
CN-114539163-B HIV-1 reverse transcriptase inhibitor and its synthesis process 复旦大学 2023-05-30 CN claimed
CN-114539163-A HIV-1 reverse transcriptase inhibitor and synthetic method thereof 复旦大学 2022-05-27 CN claimed
CN-109824602-A The synthetic method of the chloro- 2- methylthiopyrimidine of 4- 南京哈柏医药科技有限公司 2019-05-31 CN claimed
EP-4143193-B1 IMIDAZOPYRIMIDINES AS MODULATORS OF IL-17 JANSSEN PHARMACEUTICA NV (BE) 2026-04-22 EP disclosed
EP-3877382-B1 NOVEL COMPOUNDS FOR THE TREATMENT OF RESPIRATORY DISEASES TIANLI BIOTECH PTY LTD (AU) 2026-03-18 EP disclosed
US-12559496-B2 Imidazopyrimidines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2026-02-24 US disclosed
US-20260049086-A1 CDK9 INHIBITORS BAERENKRAFT THERAPEUTICS LLC (US) 2026-02-19 US disclosed
EP-3619204-B1 COMPOUNDS FOR THE TREATMENT OF RESPIRATORY DISEASES TIANLI BIOTECH PTY LTD (AU) 2025-10-01 EP disclosed
CN-115867348-B Imidazopyrimidines as IL-17 modulators 詹森药业有限公司 2025-05-06 CN disclosed
CN-113260616-B Novel compounds for the treatment of respiratory diseases 天莅生物技术有限公司 2025-05-02 CN disclosed
US-5593991-A ANTIINFLAMMATORY, CYTOKINE INHIBITOR, CYCLOOXYGENASE INHIBITOR SMITHKLINE BEECHAM CORPORATION 1997-01-14 US disclosed
US-5593992-A CYTOKINE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1997-01-14 US disclosed
WO-1996040143-A1 IMIDAZOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1996-12-19 WO disclosed
EP-0708768-A4 TRI-SUBSTITUTED IMIDAZOLES HAVING MULTIPLE THERAPEUTIC PROPERTIES SMITHKLINE BEECHAM CORP (US) 1996-08-21 EP disclosed
CN-1129447-A Trisubstituted imidazoles having multiple therapeutic effects SMITHKLINE BEECHAM CORP (US) 1996-08-21 CN disclosed
WO-1996021452-A1 CERTAIN 1,4,5-TRI-SUBSTITUTED IMIDAZOLE COMPOUNDS USEFUL AS CYTOKINE SMITHKLINE BEECHAM CORPORATION (US) 1996-07-18 WO disclosed
EP-0708768-A1 TRI-SUBSTITUTED IMIDAZOLES HAVING MULTIPLE THERAPEUTIC PROPERTIES SMITHKLINE BEECHAM CORPORATION (US) 1996-05-01 EP disclosed
WO-1995002591-A1 TRI-SUBSTITUTED IMIDAZOLES HAVING MULTIPLE THERAPEUTIC PROPERTIES SMITHKLINE BEECHAM CORPORATION (US) 1995-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260049086-A1 CDK9 INHIBITORS CDK9, CDK6, CDK19 KMT2A 834/4885MEN1 3655/4885NPC1 2438/4885
US-12559496-B2 Imidazopyrimidines as modulators of IL-17 IL17A, IL2, IL23R KMT2A 3063/4885MEN1 2259/4885NPC1 291/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.