SCHEMBL18808331

SCHEMBL18808331

CNc1ccc(C(=O)Nc2ccc(F)c(F)c2)cc1C=N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
MAOB P27338 4/20 0.50
MAOA P21397 1/20 0.50
LMNA P02545 3/20 0.49
CASP3 P42574 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
KCNQ3 O43525 5/20 0.47
KCNQ2 O43526 5/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
MEN1 O00255 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
KCNE1 P15382 1/20 0.44
KCNQ1 P51787 1/20 0.44
HTR2B P41595 1/20 0.44
KCNQ5 Q9NR82 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18808492 0.90 KCNQ3 (0.43) NPC1RAB9AMAOBMAOALMNA
SCHEMBL18808350 0.89 NPC1 (0.54) NPC1RAB9AMAOBMAOALMNA
SCHEMBL18808347 0.82 NPC1 (0.61) NPC1RAB9AMAOBMAOALMNA
SCHEMBL18808333 0.82 NPC1 (0.54) NPC1RAB9AMAOBMAOALMNA
SCHEMBL22453429 0.78 LRRK2 (0.42) NPC1RAB9AMEN1MAPTKMT2A
SCHEMBL21146669 0.77 RAB9A (0.60) NPC1RAB9AMAOBMAOALMNA
SCHEMBL22453825 0.74 HDAC3 (0.45) NPC1RAB9AMAPTKMT2A
SCHEMBL17465718 0.74 NPC1 (0.64) NPC1RAB9AMAOBMAOALMNA
SCHEMBL19936703 0.73 HCAR3 (0.51) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL22453907 0.73 ABCB1 (0.40) NPC1RAB9AMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964219-B1 SUBSTITUTED INDAZOLE OR INDOLE DERIVATIVES AS IN VITRO MAO-B INHIBITORS NTZ LAB LTD (BG) 2017-05-03 EP disclosed