SCHEMBL21574736

SCHEMBL21574736

BC(=C)C(C=C)Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.39
TAAR1 Q96RJ0 1/20 0.37
PPARG P37231 3/20 0.36
PPARA Q07869 3/20 0.36
ORAI1 Q96D31 1/20 0.35
ORAI2 Q96SN7 1/20 0.35
ORAI3 Q9BRQ5 1/20 0.35
TRPV6 Q9H1D0 1/20 0.35
TGM2 P21980 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
EPHX2 P34913 1/20 0.34
TEAD1 P28347 2/20 0.33
SRD5A2 P31213 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21076020 0.81 PPARG (0.38) IDO1TAAR1PPARGPPARANPC1
SCHEMBL21573071 0.80 HRH3 (0.37) TAAR1PPARGPPARANPC1RAB9A
SCHEMBL21075947 0.77 TAAR1 (0.45) IDO1TAAR1PPARGPPARAORAI1
SCHEMBL18856419 0.73 TP53 (0.35)
SCHEMBL7435082 0.73 TAAR1 (0.46) IDO1TAAR1NPC1RAB9AALDH1A1
SCHEMBL21538871 0.67 HTR2A (0.55) IDO1TAAR1MAOB
SCHEMBL24202494 0.67 CPA1 (0.41) TAAR1PPARGPPARA
SCHEMBL31435841 0.66 HSD11B1 (0.50) IDO1TAAR1PPARGPPARA
SCHEMBL31435844 0.66 HSD11B1 (0.50) IDO1TAAR1PPARGPPARA
SCHEMBL16868329 0.66 ALDH1A1 (0.47) IDO1TAAR1PPARGPPARANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057951-B1 METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T JANSSEN PHARMACEUTICA NV (BE) 2019-11-20 EP disclosed