SCHEMBL188597

SCHEMBL188597

O=NNC(=O)N(Cl)Cl

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257806 0.73 ALDH1A1 (0.32)
SCHEMBL609663 0.71
SCHEMBL28237964 0.67 ALDH1A1 (0.33)
SCHEMBL250276 0.67 ALDH1A1 (0.42)
SCHEMBL2465792 0.67 ALDH1A1 (0.30)
SCHEMBL22616909 0.65 LMNA (0.37)
SCHEMBL3197195 0.65
SCHEMBL2347991 0.64 CA12 (0.32)
SCHEMBL3359802 0.63
SCHEMBL7644031 0.62 TSHR (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 339 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150342165-A1 HUMANIZED MOUSE AND METHODS OF USING THE SAME CITY OF HOPE 2015-12-03 US claimed
EP-2538944-B1 COMPOUND FOR TREATING BRAIN CANCER NIIKI PHARMA INC (US) 2014-10-22 EP claimed
US-20120040914-A1 ENHANCING EFFECTIVENESS OF GLIAL CANCER THERAPIES UNIVERSITY OF NORTH TEXAS HEALTH SCIENCE CENTER AT FORT WORTH (US) 2012-02-16 US claimed
US-7858659-B2 Redox therapy for tumors HOFFMAN ARNOLD 2010-12-28 US claimed
US-20260130855-A1 GAMMA POLYGLUTAMATED ANTIFOLATES AND USES THEREOF L E A F HOLDINGS GROUP LLC (US) 2026-05-14 US disclosed
US-12622874-B2 Trans-crocetin compositions and treatment regimens L.E.A.F. HOLDINGS GROUP LLC (US) 2026-05-12 US disclosed
US-20260103694-A1 TARGETED GENE INSERTION FOR IMPROVED IMMUNE CELLS THERAPY CELLECTIS (FR) 2026-04-16 US disclosed
US-20260053806-A1 GAMMA POLYGLUTAMATED METHOTREXATE AND USES THEREOF L E A F HOLDINGS GROUP LLC (US) 2026-02-26 US disclosed
US-20260048054-A1 ALPHA POLYGLUTAMATED TETRAHYDROFOLATES AND USES THEREOF L E A F HOLDINGS GROUP LLC (US) 2026-02-19 US disclosed
US-20260014079-A1 CAROTENOID COMPOSITIONS AND USES THEREOF L E A F HOLDINGS GROUP LLC (US) 2026-01-15 US disclosed
EP-3706801-B1 PLATINUM COMPLEXES AND USES THEREOF L E A F HOLDINGS GROUP LLC (US) 2026-01-14 EP disclosed
EP-4667017-A2 CAROTENOID COMPOSITIONS AND USES THEREOF L.E.A.F Holdings Group LLC (US) 2025-12-24 EP disclosed
US-6300458-B1 High molecular weight polymers and copolymers of BHMDO for biomedical application VANDENBERG, DAVID J 2001-10-09 US disclosed
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed
US-5380759-A Methyl N-[6-(3,4,5-trimethoxybenzloxy)imidazo[1,2-b]pyridazin-2-zyl]carbamate used to treat leukemia BURROUGHS WELLCOME CO. (US) 1995-01-10 US disclosed
US-5371219-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1994-12-06 US disclosed
EP-0305093-B1 Imidazo(1,2-b)pyridazine derivatives WELLCOME FOUND (GB) 1994-04-06 EP disclosed
US-5091531-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1992-02-25 US disclosed
EP-0305093-A1 Imidazo(1,2-b)pyridazine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1989-03-01 EP disclosed