SCHEMBL188906

SCHEMBL188906

CN(C)C(CCO)c1ccc(N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.38
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
CHRNA4 P43681 2/20 0.38
ALDH1A1 P00352 4/20 0.35
TDP1 Q9NUW8 4/20 0.35
CYP3A4 P08684 2/20 0.35
MAPK1 P28482 2/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
OPRK1 P41145 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
PSMD14 O00487 1/20 0.32
TSHR P16473 1/20 0.32
RECQL P46063 1/20 0.32
GFER P55789 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
PHLPP2 Q6ZVD8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529486 0.84 ALDH1A1 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL9613800 0.81 AOC3 (0.44) CHRNB2CHRNB4CHRNA3CHRNA4TDP1
SCHEMBL4739377 0.81 AOC3 (0.44) CHRNB2CHRNB4CHRNA3CHRNA4OPRK1
SCHEMBL9995387 0.80 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL12071516 0.80 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL28144242 0.80 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL5398515 0.80 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL28144244 0.80 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
Hydrochloric Acid SCHEMBL17710458 0.78 CHRNB2 (0.54) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
Bromide SCHEMBL28176004 0.78 CHRNB2 (0.54) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401281-A1 PYRIMIDOPYRIMIDOINDAZOLE DERIVATIVE MSD K.K. (JP) 2012-01-04 EP disclosed
WO-2010098367-A1 PYRIMIDOPYRIMIDOINDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-09-02 WO disclosed