SCHEMBL529486

SCHEMBL529486

CN(C)C(CO)c1ccc(N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
CYP3A4 P08684 3/20 0.38
TDP1 Q9NUW8 3/20 0.38
MAPK1 P28482 2/20 0.38
ALOX15 P16050 2/20 0.38
TP53 P04637 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.34
PSMD14 O00487 1/20 0.34
TSHR P16473 1/20 0.34
RECQL P46063 1/20 0.34
GFER P55789 1/20 0.34
OPRK1 P41145 1/20 0.34
NOS3 P29474 3/20 0.33
NOS1 P29475 3/20 0.33
NOS2 P35228 3/20 0.33
KMT2A Q03164 2/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL188906 0.84 CHRNB2 (0.38) ALDH1A1CYP3A4TDP1MAPK1ALOX15
SCHEMBL10915673 0.79 PYCR1 (0.44) KMT2AMEN1
SCHEMBL14003539 0.79 AOC3 (0.42) ALDH1A1CYP3A4TDP1MAPK1ALOX15
SCHEMBL864654 0.79 AOC3 (0.42) ALDH1A1CYP3A4TDP1MAPK1ALOX15
SCHEMBL817422 0.78 KDM4E (0.52) ALDH1A1TDP1CHRNB2CHRNB4CHRNA3
SCHEMBL1206432 0.78 KDM4E (0.52) ALDH1A1TDP1CHRNB2CHRNB4CHRNA3
SCHEMBL1205734 0.78 KDM4E (0.52) ALDH1A1TDP1CHRNB2CHRNB4CHRNA3
SCHEMBL11488424 0.75 GRIA4 (0.41) ALDH1A1CYP3A4TDP1MAPK1ALOX15
SCHEMBL529767 0.72 TSHR (0.51) ALDH1A1CYP3A4TDP1MAPK1L3MBTL1
SCHEMBL3872917 0.72 ALDH1A1 (0.31) ALDH1A1CYP3A4ALOX15CA3THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed