SCHEMBL18894012

SCHEMBL18894012

Oc1c(Cl)cc(C(F)(F)F)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP3A4 P08684 3/20 0.43
TSHR P16473 3/20 0.43
RECQL P46063 3/20 0.43
HSD17B10 Q99714 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
ALOX15 P16050 2/20 0.43
ALOX12 P18054 2/20 0.43
HPGD P15428 1/20 0.43
CASP1 P29466 1/20 0.43
HIF1A Q16665 1/20 0.43
PDE2A O00408 1/20 0.38
ERN1 O75460 1/20 0.37
CHEK1 O14757 1/20 0.37
DAPK3 O43293 1/20 0.37
RET P07949 1/20 0.37
PDGFRB P09619 1/20 0.37
PIM1 P11309 1/20 0.37
PDGFRA P16234 1/20 0.37
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5600053 0.84 ALDH1A1 (0.50) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL10699329 0.84 TSHR (0.58) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL814586 0.79 TSHR (0.54) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL1068524 0.79 TSHR (0.72) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL4868822 0.78 TSHR (0.46) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL12635966 0.77 PDE2A (0.43) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL8773859 0.77 PDE2A (0.39) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL20974042 0.77 TSHR (0.50) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL15729337 0.77 TSHR (0.45) ALDH1A1CYP3A4TSHRRECQLHSD17B10
SCHEMBL10680627 0.77 GABRB3 (0.36) ALDH1A1CYP3A4TSHRRECQLTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3636651-A1 HEXAHYDROPYRAZINOBENZ- OR -PYRIDO-OXAZEPINES CARRYING AN OXYGEN-CONTAINING SUBSTITUENT AND USE THEREOF IN THE TREATMENT OF 5-HT2C-DEPENDENT DISORDERS AbbVie Deutschland GmbH & Co. KG (DE) 2020-04-15 EP disclosed
US-20180339996-A1 HEXAHYDROPYRAZINOBENZ- OR -PYRIDO-OXAZEPINES CARRYING AN OXYGEN-CONTAINING SUBSTITUENT AND USE THEREOF IN THE TREATMENT OF 5-HT2C-DEPENDENT DISORDERS AbbVie Deutschland GmbH & Co. KG (DE) 2018-11-29 US disclosed
EP-3380483-A1 HEXAHYDROPYRAZINOBENZ- OR -PYRIDO-OXAZEPINES CARRYING AN OXYGEN-CONTAINING SUBSTITUENT AND USE THEREOF IN THE TREATMENT OF 5-HT2C-DEPENDENT DISORDERS Abbvie Deutschland GmbH & Co. KG (DE) 2018-10-03 EP disclosed
WO-2017089458-A1 HEXAHYDROPYRAZINOBENZ- OR -PYRIDO-OXAZEPINES CARRYING AN OXYGEN-CONTAINING SUBSTITUENT AND USE THEREOF IN THE TREATMENT OF 5-HT2C-DEPENDENT DISORDERS AbbVie Deutschland GmbH & Co. KG (DE) 2017-06-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180339996-A1 HEXAHYDROPYRAZINOBENZ- OR -PYRIDO-OXAZEPINES CARRYING AN OXYGEN-CONTAINING SUBSTITUENT AND USE THEREOF IN THE TREATMENT OF 5-HT2C-DEPENDENT DISORDERS HTR2C, HTR2A, HTR5A ALDH1A1 821/4885CYP3A4 350/4885TSHR 659/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.